SCHEMBL856116

SCHEMBL856116

CC1(C)CCc2nc(CN(C(=O)OCc3ccccc3)C3CCC3)nc(Cl)c2C1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 3/20 0.40
ACHE P22303 6/20 0.37
SIGMAR1 Q99720 1/20 0.37
CCR5 P51681 6/20 0.37
HTR2A P28223 1/20 0.36
ENPP2 Q13822 1/20 0.36
AGER Q15109 1/20 0.35
RORC P51449 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL857343 0.99 PTGDR2 (0.41) PTGDR2ACHESIGMAR1CCR5HTR2A
SCHEMBL856161 0.85 ACHE (0.38) PTGDR2ACHERORC
SCHEMBL856425 0.84 ACHE (0.36) ACHESIGMAR1RORC
SCHEMBL3723441 0.83 ACHE (0.35) ACHEAGER
SCHEMBL857298 0.83 ACHE (0.35) PTGDR2ACHERORC
SCHEMBL3717335 0.82 AGER (0.34) ACHEAGER
SCHEMBL856242 0.82 ACHE (0.35) ACHERORC
SCHEMBL858893 0.76 TP53 (0.35) ACHE
SCHEMBL856154 0.74 AADAT (0.43) SIGMAR1
SCHEMBL856612 0.74 AADAT (0.43) SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2432779-A1 BENZOXAZEPINES BASED P13K/MT0R INHIBITORS AGAINST PROLIFERATIVE DISEASES Exelixis, Inc. (US) 2012-03-28 EP disclosed