SCHEMBL856242

SCHEMBL856242

CC1(C)CCc2nc(CN(CC(F)F)C(=O)OCc3ccccc3)nc(Cl)c2C1

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ACHE P22303 9/20 0.35
MAPK1 P28482 1/20 0.33
ALDH1A1 P00352 1/20 0.32
RORC P51449 3/20 0.32
DDB1 Q16531 1/20 0.31
CRBN Q96SW2 1/20 0.31
CCR1 P32246 1/20 0.31
CCR6 P51684 1/20 0.31
PAX8 Q06710 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL856161 0.89 ACHE (0.38) ACHEMAPK1ALDH1A1RORC
SCHEMBL857298 0.89 ACHE (0.35) ACHEMAPK1RORCDDB1CRBN
SCHEMBL856425 0.85 ACHE (0.36) ACHEMAPK1ALDH1A1RORC
SCHEMBL856116 0.82 PTGDR2 (0.40) ACHERORC
SCHEMBL857343 0.81 PTGDR2 (0.41) ACHE
SCHEMBL857154 0.68 PDK1 (0.35) MAPK1
SCHEMBL3723441 0.68 ACHE (0.35) ACHEALDH1A1
SCHEMBL856626 0.68 AADAT (0.43)
SCHEMBL858958 0.66 PDK1 (0.33) ACHEMAPK1
SCHEMBL856424 0.66 ACHE (0.37) ACHEMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2432779-A1 BENZOXAZEPINES BASED P13K/MT0R INHIBITORS AGAINST PROLIFERATIVE DISEASES Exelixis, Inc. (US) 2012-03-28 EP disclosed