SCHEMBL8561422

SCHEMBL8561422

COC(=O)O[C@@]1(NC(=O)OC(C)(C)C)CCc2cccc(Oc3ccc([N+](=O)[O-])cc3C(=O)OCc3ccccc3)c2C1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSV O60911 1/20 0.36
CTSL P07711 1/20 0.36
MAPT P10636 1/20 0.36
ITGA4 P13612 1/20 0.36
ITGB7 P26010 1/20 0.36
PDE1C Q14123 1/20 0.35
LMNA P02545 3/20 0.35
ALDH1A1 P00352 1/20 0.35
RAB9A P51151 3/20 0.34
PAX8 Q06710 1/20 0.34
MITF O75030 1/20 0.34
KMT2A Q03164 4/20 0.34
CYP19A1 P11511 1/20 0.34
NPC1 O15118 1/20 0.34
HTT P42858 2/20 0.34
POLB P06746 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
ACHE P22303 1/20 0.34
MEN1 O00255 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8567143 0.90 CA1 (0.39) CTSLMAPTALDH1A1KMT2APOLB
SCHEMBL8575729 0.90 CA1 (0.39) CTSLMAPTALDH1A1KMT2APOLB
SCHEMBL8845255 0.89 CTSV (0.38) CTSVCTSLMAPTITGA4ITGB7
SCHEMBL8997699 0.83 CA1 (0.36) ALDH1A1RAB9ANPC1HTTPOLB
SCHEMBL8560808 0.81 SYK (0.35) CTSLMAPTLMNAALDH1A1CA1
SCHEMBL8574453 0.80 CA1 (0.35) CTSLMAPTALDH1A1CA1CA2
SCHEMBL8997600 0.80 SYK (0.40) MAPTITGA4ITGB7LMNAALDH1A1
SCHEMBL8573147 0.79 CYP3A4 (0.37) MAPTALDH1A1
SCHEMBL8997778 0.79 MEN1 (0.40) ALDH1A1RAB9AKMT2ANPC1HTT
SCHEMBL8997648 0.79 SYK (0.38) CTSLCA1CA2ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640618-B1 Tetrahydronaphthalene-peptide derivatives HOFFMANN LA ROCHE (CH) 1999-10-20 EP disclosed
EP-0640618-A1 Tetrahydronaphthalene-peptide derivatives F. HOFFMANN-LA ROCHE AG (CH) 1995-03-01 EP disclosed