SCHEMBL8562834

SCHEMBL8562834

Cc1nc(Br)n(COCc2ccccc2)c1Sc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.44
VCP P55072 2/20 0.36
TSHR P16473 2/20 0.35
USP2 O75604 1/20 0.34
MAPK1 P28482 1/20 0.34
L3MBTL1 Q9Y468 2/20 0.34
CYP2C9 P11712 2/20 0.33
CYP2C19 P33261 2/20 0.33
GCK P35557 1/20 0.32
SMN1; SMN2 Q16637 3/20 0.32
STAT3 P40763 1/20 0.32
HTT P42858 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
POLB P06746 1/20 0.32
ATP4A P20648 2/20 0.31
ATP4B P51164 2/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9051616 0.87 ALDH1A1 (0.40) ALDH1A1VCPTSHRUSP2MAPK1
SCHEMBL9050612 0.86 ALDH1A1 (0.40) ALDH1A1VCPTSHRMAPK1L3MBTL1
SCHEMBL8567515 0.86 VCP (0.41) ALDH1A1VCPTSHRL3MBTL1CYP2C9
SCHEMBL8568227 0.85 ALDH1A1 (0.39) ALDH1A1VCPTSHRMAPK1L3MBTL1
SCHEMBL8562572 0.84 ALDH1A1 (0.38) ALDH1A1VCPTSHRL3MBTL1CYP2C9
Hydrochloric Acid SCHEMBL8563542 0.81 ALDH1A1 (0.39) ALDH1A1VCPTSHRL3MBTL1CYP2C9
SCHEMBL8567357 0.80 ALDH1A1 (0.38) ALDH1A1TSHRL3MBTL1CYP2C9CYP2C19
SCHEMBL8567153 0.78 CSNK1D (0.42) ALDH1A1TSHRMAPK1L3MBTL1SMN1; SMN2
SCHEMBL8560120 0.75 ALDH1A1 (0.38) ALDH1A1VCPTSHRL3MBTL1CYP2C9
Nitric Acid SCHEMBL8566793 0.73 ALDH1A1 (0.39) ALDH1A1TSHRMAPK1L3MBTL1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0552060-B1 Imidazole derivatives having anti-HIV activity SHIONOGI & CO (JP) 1998-11-18 EP disclosed
EP-0700911-A1 Imidazole derivatives having anti-HIV activity SHIONOGI & CO., LTD. (JP) 1996-03-13 EP disclosed
US-5472965-A Useful for treatment of retrovirus infections; less toxic SHIONOGI & CO., LTD. (JP) 1995-12-05 US disclosed
US-5326780-A Acquired immunodeficiency syndrome SHIONOGI & CO., LTD. (JP) 1994-07-05 US disclosed
EP-0552060-A1 Imidazole derivatives having anti-HIV activity SHIONOGI & CO., LTD. (JP) 1993-07-21 EP disclosed