SCHEMBL8562850

SCHEMBL8562850

CC(C)(C)OC(=O)c1ccc(CCCn2ccc(N)c2C#N)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP4A11 Q02928 2/20 0.35
CA12 O43570 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA9 Q16790 1/20 0.35
CA14 Q9ULX7 1/20 0.35
SIRT2 Q8IXJ6 1/20 0.35
SIRT1 Q96EB6 1/20 0.35
EP300 Q09472 3/20 0.35
CYP4F2 P78329 1/20 0.34
NR3C2 P08235 2/20 0.33
HDAC3 O15379 2/20 0.32
HDAC4 P56524 2/20 0.32
HDAC1 Q13547 2/20 0.32
HDAC7 Q8WUI4 2/20 0.32
HDAC2 Q92769 2/20 0.32
HDAC10 Q969S8 2/20 0.32
HDAC11 Q96DB2 2/20 0.32
HDAC8 Q9BY41 2/20 0.32
HDAC6 Q9UBN7 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8564883 0.81 CA12 (0.34) CA12CA1CA2CA9CA14
SCHEMBL8567733 0.80 CRHBP (0.41) CYP4A11CA12CA1CA2CA9
SCHEMBL8569504 0.80 NR3C2 (0.34) CA12CA1CA2CA9CA14
SCHEMBL8569300 0.80 ATIC (0.33) NR3C2
SCHEMBL8565003 0.80 CA12 (0.36) CA12CA1CA2CA9CA14
SCHEMBL8567809 0.79 CA12 (0.36) CA12CA1CA2CA9CA14
SCHEMBL8567806 0.79 CA12 (0.36) CA12CA1CA2CA9CA14
SCHEMBL8563771 0.74 TLR7 (0.45) CA12CA1CA2CA9CA14
SCHEMBL9001785 0.73 TLR7 (0.44) CYP4A11CA12CA1CA2CA9
SCHEMBL31688879 0.71 CYP4A11 (0.49) CYP4A11CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530579-B1 Condensed pyrimidine derivatives antitumor agents EISAI CO LTD (JP) 1998-11-11 EP disclosed
US-5688800-A ANTITUMOR AGENTS EISAI CO., LTD. (JP) 1997-11-18 US disclosed
US-5554615-A ANTITUMOR EISAI CO., LTD. (JP) 1996-09-10 US disclosed
EP-0530579-A1 Condensed pyrimidine derivatives antitumor agents Eisai Co., Ltd. (JP) 1993-03-10 EP disclosed