SCHEMBL8569300

SCHEMBL8569300

CC(C)(C)OC(=O)c1ccc(CCCn2ccc(N)c2C#N)s1

nearest known ligand 0.33

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ATIC P31939 3/20 0.33
SHMT1 P34896 3/20 0.33
SHMT2 P34897 3/20 0.33
NR3C2 P08235 2/20 0.32
HPGD P15428 1/20 0.32
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
PRNP P04156 1/20 0.31
RECQL P46063 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31
GART P22102 2/20 0.31
POLB P06746 1/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8562850 0.80 CYP4A11 (0.35) NR3C2
SCHEMBL8564673 0.75 ATIC (0.43) ATICSHMT1SHMT2HPGDALDH1A1
SCHEMBL5050275 0.73 HPGD (0.42) HPGDALDH1A1LMNAPRNPRECQL
Hydrochloric Acid SCHEMBL5724631 0.72 HPGD (0.41) HPGDALDH1A1LMNAPRNPRECQL
Hydrochloric Acid SCHEMBL2413233 0.72 HPGD (0.40) HPGDALDH1A1LMNAPRNPRECQL
SCHEMBL8570240 0.72 HPGD (0.43) HPGDALDH1A1LMNAPRNPRECQL
SCHEMBL21199747 0.71 POLB (0.46) HPGDALDH1A1LMNAPRNPRECQL
SCHEMBL8982459 0.71 HPGD (0.45) HPGDALDH1A1LMNAPRNPRECQL
SCHEMBL8564545 0.71 HPGD (0.45) HPGDALDH1A1LMNAPRNPRECQL
SCHEMBL8564883 0.70 CA12 (0.34) NR3C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530579-B1 Condensed pyrimidine derivatives antitumor agents EISAI CO LTD (JP) 1998-11-11 EP disclosed
US-5688800-A ANTITUMOR AGENTS EISAI CO., LTD. (JP) 1997-11-18 US disclosed
US-5554615-A ANTITUMOR EISAI CO., LTD. (JP) 1996-09-10 US disclosed
EP-0530579-A1 Condensed pyrimidine derivatives antitumor agents Eisai Co., Ltd. (JP) 1993-03-10 EP disclosed