SCHEMBL8563771

SCHEMBL8563771

CC(C)(C)OC(=O)c1ccc(CCCn2ccc3nc(N)nc(N)c32)cc1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TLR7 Q9NYK1 6/20 0.45
ATIC P31939 3/20 0.40
SHMT1 P34896 3/20 0.40
SHMT2 P34897 3/20 0.40
GART P22102 2/20 0.38
EP300 Q09472 4/20 0.37
F2R P25116 1/20 0.35
TLR8 Q9NR97 1/20 0.35
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
CA14 Q9ULX7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9001785 0.91 TLR7 (0.44) TLR7ATICSHMT1SHMT2GART
SCHEMBL8570678 0.88 ATIC (0.38) TLR7ATICSHMT1SHMT2GART
SCHEMBL8563902 0.84 TLR7 (0.50) TLR7ATICSHMT1SHMT2GART
SCHEMBL8571595 0.81 TLR7 (0.38) TLR7F2RCA12CA1CA2
SCHEMBL8564673 0.81 ATIC (0.43) TLR7ATICSHMT1SHMT2GART
SCHEMBL8564223 0.80 TLR7 (0.37) TLR7F2RCA12CA1CA2
SCHEMBL8564228 0.80 TLR7 (0.37) TLR7F2RCA12CA1CA2
SCHEMBL8564668 0.80 ATIC (0.48) TLR7ATICSHMT1SHMT2GART
SCHEMBL9446114 0.77 DHFR (0.46)
SCHEMBL8567733 0.74 CRHBP (0.41) EP300CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530579-B1 Condensed pyrimidine derivatives antitumor agents EISAI CO LTD (JP) 1998-11-11 EP disclosed
US-5688800-A ANTITUMOR AGENTS EISAI CO., LTD. (JP) 1997-11-18 US disclosed
US-5554615-A ANTITUMOR EISAI CO., LTD. (JP) 1996-09-10 US disclosed
EP-0530579-A1 Condensed pyrimidine derivatives antitumor agents Eisai Co., Ltd. (JP) 1993-03-10 EP disclosed