SCHEMBL8562874

SCHEMBL8562874

CC(C)(C)OC(=O)c1ccc(CNC(=O)C(Br)CCBr)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMO Q99835 1/20 0.46
SIRT2 Q8IXJ6 1/20 0.38
SIRT1 Q96EB6 1/20 0.38
NAMPT P43490 1/20 0.38
NR1H4 Q96RI1 6/20 0.38
EPHX2 P34913 6/20 0.38
GAA P10253 1/20 0.38
CA1 P00915 3/20 0.37
CA2 P00918 3/20 0.37
HDAC6 Q9UBN7 2/20 0.37
MEN1 O00255 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
KMT2A Q03164 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
CYP2D6 P10635 1/20 0.37
CA12 O43570 1/20 0.36
CA9 Q16790 1/20 0.36
CA14 Q9ULX7 1/20 0.36
HDAC3 O15379 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8563816 0.83 NAMPT (0.47) NAMPTEPHX2GAACA1CA2
SCHEMBL27520455 0.80 KMT2A (0.53) NAMPTNR1H4EPHX2MEN1KMT2A
SCHEMBL23409688 0.79 HTT (0.47) NAMPTNR1H4EPHX2GAACA1
SCHEMBL16885994 0.78 KMT2A (0.54) GAAMEN1NPC1RAB9AKMT2A
SCHEMBL8562984 0.78 ALDH1A1 (0.51) GAAMEN1NPC1RAB9AKMT2A
SCHEMBL8562987 0.78 ALDH1A1 (0.51) GAAMEN1NPC1RAB9AKMT2A
SCHEMBL6945571 0.77 HTT (0.50) NAMPTNR1H4EPHX2GAACA1
SCHEMBL10165179 0.77 NAMPT (0.56) NAMPTNR1H4EPHX2GAACA1
SCHEMBL19682558 0.77 KMT2A (0.60) NAMPTNR1H4EPHX2GAACA1
SCHEMBL1543096 0.76 MEN1 (0.54) GAAMEN1NPC1RAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1060778-C Cephalosporin derivatives HOFFMANN LA ROCHE (CH) 2001-01-17 CN disclosed
US-5804577-A ANTIBIOTICS HOFFMANN-LA ROCHE INC. (US) 1998-09-08 US disclosed