SCHEMBL8563056

SCHEMBL8563056

Cc1occc1CC(=O)Nc1ccc(C(=O)N2CCc3ccccc3-c3ccccc32)cc1

nearest known ligand 0.60

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.48
MAPT P10636 1/20 0.48
NAMPT P43490 1/20 0.47
NPC1 O15118 1/20 0.46
HPGD P15428 1/20 0.46
RAB9A P51151 1/20 0.46
KMT2A Q03164 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
AVPR1A P37288 2/20 0.45
AVPR2 P30518 3/20 0.44
LDHA P00338 1/20 0.44
LDHB P07195 1/20 0.44
OXTR P30559 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8557382 0.87 AVPR2 (0.50) NAMPTNPC1HPGDRAB9AKMT2A
SCHEMBL8563752 0.85 ALDH1A1 (0.57) ALDH1A1MAPTAVPR1AAVPR2OXTR
SCHEMBL8564664 0.83 NAMPT (0.47) NAMPTNPC1HPGDRAB9AKMT2A
SCHEMBL8561675 0.83 NAMPT (0.50) ALDH1A1NAMPTAVPR1A
SCHEMBL8558667 0.82 NAMPT (0.54) ALDH1A1MAPTNAMPTNPC1HPGD
SCHEMBL8558454 0.80 GRM1 (0.57) AVPR1AAVPR2OXTR
SCHEMBL7331304 0.77 KMT2A (0.48) KMT2AAVPR1AAVPR2
SCHEMBL8312861 0.76 AVPR1A (0.45) AVPR1AAVPR2
SCHEMBL8562680 0.76 ALDH1A1 (0.59) ALDH1A1NAMPTHPGDRAB9AAVPR1A
SCHEMBL8316301 0.76 AVPR2 (0.42) AVPR1AAVPR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640592-B1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID CO (US) 1998-12-30 EP disclosed
EP-0640592-A1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID COMPANY (US) 1995-03-01 EP disclosed