SCHEMBL8562828

SCHEMBL8562828

Cc1ccc(C)c(NC(=O)c2ccc(C(=O)N3Cc4ccccc4Cc4ccccc43)cc2)c1

nearest known ligand 0.61

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 2/20 0.49
AVPR1A P37288 2/20 0.49
LMNA P02545 2/20 0.49
RAB9A P51151 2/20 0.48
POLB P06746 2/20 0.47
KMT2A Q03164 2/20 0.47
MEN1 O00255 1/20 0.47
GAA P10253 1/20 0.47
TP53 P04637 1/20 0.47
MAPT P10636 1/20 0.47
NPC1 O15118 1/20 0.46
HPGD P15428 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
APOBEC3A P31941 1/20 0.46
APOBEC3G Q9HC16 1/20 0.46
ACHE P22303 1/20 0.45
HSD17B3 P37058 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8562097 0.92 AVPR2 (0.49) AVPR2AVPR1ALMNARAB9APOLB
SCHEMBL8562633 0.89 AVPR2 (0.55) AVPR2AVPR1ALMNARAB9APOLB
SCHEMBL8563072 0.84 SMN1; SMN2 (0.55) AVPR2AVPR1ALMNARAB9AKMT2A
SCHEMBL8558733 0.83 AVPR2 (0.65) AVPR2AVPR1A
SCHEMBL9236961 0.82 AVPR2 (0.66) AVPR2AVPR1A
SCHEMBL8557607 0.80 NPC1 (0.50) AVPR2AVPR1ARAB9APOLBGAA
SCHEMBL8558857 0.80 HPGD (0.57) RAB9AKMT2AMEN1NPC1HPGD
SCHEMBL8561645 0.79 AVPR2 (0.58) AVPR2AVPR1ARAB9ANPC1ACHE
SCHEMBL8559546 0.79 AVPR2 (0.55) AVPR2AVPR1AKMT2AMEN1ACHE
SCHEMBL8560873 0.78 ACHE (0.60) AVPR2AVPR1ARAB9AACHEHSD17B3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640592-B1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID CO (US) 1998-12-30 EP disclosed