SCHEMBL856332

SCHEMBL856332

O=C1C=C(c2cc3ccccc3[nH]2)C(=O)N1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 2/20 0.51
CHEK1 O14757 1/20 0.51
RAB9A P51151 4/20 0.49
NPC1 O15118 4/20 0.49
KDM4E B2RXH2 3/20 0.44
MAPT P10636 3/20 0.44
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
ALDH1A1 P00352 2/20 0.44
HPGD P15428 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
PRKD3 O94806 4/20 0.44
PRKCG P05129 4/20 0.44
PRKCB P05771 4/20 0.44
PRKCA P17252 4/20 0.44
PRKCH P24723 4/20 0.44
PRKCI P41743 4/20 0.44
PRKCE Q02156 4/20 0.44
PRKCQ Q04759 4/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29900484 1.00 KDR (0.51) KDRCHEK1RAB9ANPC1KDM4E
Aniline SCHEMBL27928992 0.91 RAB9A (0.45) KDRCHEK1RAB9ANPC1KDM4E
Trifluoromethanesulfonic Acid SCHEMBL7811066 0.87 KDR (0.40) KDRCHEK1RAB9ANPC1KDM4E
Imidazole SCHEMBL5232078 0.85 CYP19A1 (0.40) KDRCHEK1RAB9ANPC1KDM4E
SCHEMBL29415921 0.79 PRKD3 (0.62) KDRCHEK1RAB9ANPC1KDM4E
SCHEMBL78989 0.79 PRKD3 (0.62) KDRCHEK1RAB9ANPC1KDM4E
SCHEMBL3959789 0.77 PRKD3 (0.61) KDRCHEK1RAB9ANPC1KDM4E
SCHEMBL5454930 0.73 KDR (0.51) KDRCHEK1RAB9ANPC1KDM4E
SCHEMBL1158440 0.73 KDR (0.51) KDRCHEK1RAB9ANPC1KDM4E
SCHEMBL31055001 0.73 KDR (0.51) KDRCHEK1RAB9ANPC1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 412 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112575449-B Polypropylene non-woven fabric with antibacterial property and preparation method thereof 广州市新君发无纺布制品包装材料有限公司 2022-05-13 CN claimed
CN-112575449-A Polypropylene non-woven fabric with antibacterial property and preparation method thereof 广州市新君发无纺布制品包装材料有限公司 2021-03-30 CN claimed
US-20200385685-A1 ROBUST DIFFERENTIATION OF HUMAN PLURIPOTENT STEM CELLS INTO ENDOTHELIAL CELLS USING TRANSCRIPTION FACTOR ETV2 CHILDREN'S MEDICAL CENTER CORPORATION 2020-12-10 US claimed
CN-106188007-B A kind of 3- piperidyls -4- indolylmaleimides class compounds and its preparation and application 东华大学 2018-08-14 CN claimed
CN-108264503-A A kind of preparation method of 3- Indolylmaleimide compounds 东华大学 2018-07-10 CN claimed
CN-106188007-A A kind of 3 piperidyl 4 indolylmaleimides compounds and preparation thereof and application 东华大学 2016-12-07 CN claimed
CN-105153126-A Preparation method of bisindolyl maleimide compounds NAT UNIV DONG HWA 2015-12-16 CN claimed
CN-103998444-A Adhesive agent CANCER THERAPEUTICS CRC PTY LTD 2014-08-20 CN claimed
CN-101671329-B Indolylmaleimide compound substituted with 3-amino alcohol, preparation method and application thereof UNIV DONGHUA 2012-11-07 CN claimed
CN-101671329-A Indolylmaleimide compound substituted with 3-amino alcohol, preparation method and application thereof UNIV DONGHUA 2010-03-17 CN claimed
WO-2004083202-A1 A PROCESS FOR THE PREPARATION OF INDOLYMALEIMIDES SUVEN LIFE SCIENCES LIMITED (IN) 2004-09-30 WO claimed
EP-1441772-A2 POLYMER CONJUGATES OF PROTEIN KINASE C INHIBITORS Nektar Therapeutics Al, Corporation (US) 2004-08-04 EP claimed
US-20030143185-A1 Polymer conjugates of protein kinase C inhibitors SHEARWATER CORPORATION 2003-07-31 US claimed
WO-2003037384-A2 POLYMER CONJUGATES OF PROTEIN KINASE C INHIBITORS NEKTAR THERAPEUTICS AL, CORPORATION (US) 2003-05-08 WO claimed
EP-1224932-A1 DRUGS INHIBITING CELL DEATH SAGAMI CHEMICAL RESEARCH CENTER (JP) 2002-07-24 EP claimed
EP-0888339-A4 SYNTHESIS OF INDOLYLMALEIMIDES LILLY CO ELI (US) 2001-02-28 EP claimed
US-5919946-A REACTING AN ACTIVATED MALEIMIDE WITH AN ORGANOMETALLIC-3-INDOLE IN PRESENCE OF A PALLADIUM TRANSITION METAL CATALYST ELI LILLY AND COMPANY (US) 1999-07-06 US claimed
US-5859261-A PROTEIN KINASE INHIBITORS ELI LILLY AND COMPANY (US) 1999-01-12 US claimed
EP-0888339-A1 SYNTHESIS OF INDOLYLMALEIMIDES ELI LILLY AND COMPANY (US) 1999-01-07 EP claimed
WO-1997034890-A1 SYNTHESIS OF INDOLYLMALEIMIDES ELI LILLY AND COMPANY (US) 1997-09-25 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030143185-A1 Polymer conjugates of protein kinase C inhibitors PRKCH, PRKCI, PRKCA KDR 1868/4885CHEK1 503/4885RAB9A 3147/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.