SCHEMBL29415921

SCHEMBL29415921

O=C1NC(=O)C(c2cc3ccccc3[nH]2)=C1c1cc2ccccc2[nH]1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKD3 O94806 5/20 0.62
PRKCG P05129 5/20 0.62
PRKCB P05771 5/20 0.62
PRKCA P17252 5/20 0.62
PRKCH P24723 5/20 0.62
PRKCI P41743 5/20 0.62
PRKCE Q02156 5/20 0.62
PRKCQ Q04759 5/20 0.62
PRKCZ Q05513 5/20 0.62
PRKCD Q05655 5/20 0.62
PRKD1 Q15139 5/20 0.62
PRKACA P17612 2/20 0.62
PRKACG P22612 2/20 0.62
PRKACB P22694 2/20 0.62
KDR P35968 2/20 0.58
CHEK1 O14757 1/20 0.58
RAB9A P51151 4/20 0.55
NPC1 O15118 4/20 0.55
KDM4E B2RXH2 3/20 0.49
MAPT P10636 3/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL78989 1.00 PRKD3 (0.62) PRKD3PRKCGPRKCBPRKCAPRKCH
SCHEMBL3959789 0.98 PRKD3 (0.61) PRKD3PRKCGPRKCBPRKCAPRKCH
SCHEMBL3148480 0.92 NPC1 (0.61) PRKD3PRKCGPRKCBPRKCAPRKCH
SCHEMBL31615194 0.92 NPC1 (0.61) PRKD3PRKCGPRKCBPRKCAPRKCH
SCHEMBL3908537 0.88 PRKD3 (0.59) PRKD3PRKCGPRKCBPRKCAPRKCH
SCHEMBL6417753 0.88 PRKD3 (0.56) PRKD3PRKCGPRKCBPRKCAPRKCH
SCHEMBL12424814 0.85 KDR (0.54) PRKD3PRKCGPRKCBPRKCAPRKCH
SCHEMBL2986726 0.85 PRKD3 (0.53) PRKD3PRKCGPRKCBPRKCAPRKCH
SCHEMBL3257968 0.84 PRKD3 (0.49) PRKD3PRKCGPRKCBPRKCAPRKCH
SCHEMBL15758300 0.83 PRKCB (0.64) PRKD3PRKCGPRKCBPRKCAPRKCH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260042778-A1 Polymorphs of N-Desmethyl Ruboxistaurin and Salts Thereof 4M THERAPEUTICS INC. (US) 2026-02-12 US disclosed
EP-4654966-A1 METHODS AND COMPOSITIONS FOR TREATMENT OF OBESITY AND DISEASES ASSOCIATED WITH FAT CELL ENLARGEMENT MELLICELL, INC. (US) 2025-12-03 EP disclosed
US-20250228821-A1 N-DESMETHYL RUBOXISTAURIN AS A KINASE INHIBITOR 4M THERAPEUTICS INC. (US) 2025-07-17 US disclosed
EP-4504178-A1 N-DESMETHYL RUBOXISTAURIN AS KINASE INHIBITOR 4M THERAPEUTICS INC. (US) 2025-02-12 EP disclosed
WO-2024220957-A1 POLYMORPHS OF N-DESMETHYL RUBOXISTAURIN AND SALTS THEREOF 4M THERAPEUTICS INC. (US) 2024-10-24 WO disclosed
WO-2024159211-A1 METHODS AND COMPOSITIONS FOR TREATMENT OF OBESITY AND DISEASES ASSOCIATED WITH FAT CELL ENLARGEMENT MELLICELL, INC. (US) 2024-08-02 WO disclosed
CN-110551678-B SC-beta cells, compositions and methods for producing the same 哈佛学院校长同事会 2024-02-20 CN disclosed
WO-2023192984-A1 N-DESMETHYL RUBOXISTAURIN AS KINASE INHIBITOR 4M THERAPEUTICS INC. (US) 2023-10-05 WO disclosed
US-20230285357-A1 COMPOSITIONS AND METHODS FOR TRANSDIFFERENTIATING CELLS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2023-09-14 US disclosed
US-20220244263-A1 METHODS FOR TREATING SMALL CELL NEUROENDOCRINE AND RELATED CANCERS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2022-08-04 US disclosed
US-20220081412-A1 QUINOLINYL-PYRAZINE-CARBOXAMIDE COMPOUNDS AND USES THEREOF THE REGENTS OF THE UNIVERSITY OF MICHIGAN 2022-03-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220081412-A1 QUINOLINYL-PYRAZINE-CARBOXAMIDE COMPOUNDS AND USES THEREOF HMGB3, HCCS, ACACA PRKD3 2027/4885PRKCG 1702/4885PRKCB 1249/4885
US-20260042778-A1 Polymorphs of N-Desmethyl Ruboxistaurin and Salts Thereof GSK3B, GSK3A, LRRK2 PRKD3 30/4885PRKCG 117/4885PRKCB 41/4885
US-20250228821-A1 N-DESMETHYL RUBOXISTAURIN AS A KINASE INHIBITOR GSK3B, GSK3A, GSKIP PRKD3 47/4885PRKCG 824/4885PRKCB 379/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.