SCHEMBL8563394

SCHEMBL8563394

COc1ccc(C(=O)Nc2ccc(C(=O)N3c4ccccc4CNc4ccccc43)cc2)c(OC)c1

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.50
RAB9A P51151 3/20 0.50
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
ALDH1A1 P00352 1/20 0.46
NAMPT P43490 3/20 0.45
KDR P35968 1/20 0.45
TP53 P04637 1/20 0.44
MAPT P10636 1/20 0.44
KDM4E B2RXH2 1/20 0.43
LMNA P02545 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
AVPR2 P30518 2/20 0.42
AVPR1A P37288 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8563279 0.90 AVPR2 (0.48) MEN1KMT2AALDH1A1AVPR2AVPR1A
SCHEMBL8557610 0.90 MAPT (0.52) NPC1RAB9AKMT2AALDH1A1TP53
SCHEMBL8563047 0.84 AVPR1A (0.51) RAB9AKMT2ANAMPTMAPTKDM4E
SCHEMBL8559901 0.81 AVPR2 (0.63) AVPR2AVPR1A
SCHEMBL8557927 0.81 AVPR2 (0.51) AVPR2AVPR1A
SCHEMBL8561948 0.81 AVPR2 (0.51) AVPR2AVPR1A
SCHEMBL8556562 0.80 KCNK3 (0.44) NAMPTAVPR2AVPR1A
SCHEMBL8563496 0.80 AVPR2 (0.56) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL8557883 0.79 MEN1 (0.50) NPC1RAB9AMEN1KMT2AALDH1A1
SCHEMBL8560617 0.79 AVPR1A (0.49) RAB9AMAPTLMNASMN1; SMN2AVPR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640592-B1 N-acylated tricyclic azaheterorings useful as vasopressin antagonists AMERICAN CYANAMID CO (US) 1998-12-30 EP disclosed