SCHEMBL8564223

SCHEMBL8564223

C/C=C(\Cn1ccc2nc(N)nc(N)c21)c1ccc(C(=O)OC(C)(C)C)cc1

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TLR7 Q9NYK1 4/20 0.37
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34
CA14 Q9ULX7 1/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
GLA P06280 1/20 0.34
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
THRB P10828 1/20 0.34
HPGD P15428 1/20 0.34
HIF1A Q16665 1/20 0.34
DHFR P00374 1/20 0.34
ABCG2 Q9UNQ0 1/20 0.32
F2R P25116 1/20 0.32
SLC2A1 P11166 1/20 0.31
F11 P03951 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8564228 1.00 TLR7 (0.37) TLR7CA12CA1CA2CA9
SCHEMBL8571595 0.86 TLR7 (0.38) TLR7CA12CA1CA2CA9
SCHEMBL8563771 0.80 TLR7 (0.45) TLR7CA12CA1CA2CA9
SCHEMBL8564762 0.75 SLC2A1 (0.34) TLR7CA12CA1CA2CA9
SCHEMBL8567806 0.73 CA12 (0.36) CA12CA1CA2CA9CA14
SCHEMBL8567809 0.73 CA12 (0.36) CA12CA1CA2CA9CA14
SCHEMBL8566860 0.73 CA12 (0.34) CA12CA1CA2CA9CA14
SCHEMBL9001785 0.71 TLR7 (0.44) TLR7CA12CA1CA2CA9
SCHEMBL8564673 0.70 ATIC (0.43) TLR7KDM4EALDH1A1GLAGAA
SCHEMBL8570678 0.69 ATIC (0.38) TLR7CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530579-B1 Condensed pyrimidine derivatives antitumor agents EISAI CO LTD (JP) 1998-11-11 EP disclosed
US-5554615-A ANTITUMOR EISAI CO., LTD. (JP) 1996-09-10 US disclosed
EP-0530579-A1 Condensed pyrimidine derivatives antitumor agents Eisai Co., Ltd. (JP) 1993-03-10 EP disclosed