SCHEMBL8564762

SCHEMBL8564762

CCC(c1ccc(C(=O)OC(C)(C)C)cc1)C(C)n1ccc2nc(N)nc(N)c21

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 3/20 0.34
DHFR P00374 4/20 0.33
KDM4E B2RXH2 2/20 0.32
ALDH1A1 P00352 2/20 0.32
GLA P06280 2/20 0.32
GAA P10253 2/20 0.32
MAPT P10636 2/20 0.32
HPGD P15428 2/20 0.32
HIF1A Q16665 2/20 0.32
THRB P10828 1/20 0.32
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA9 Q16790 1/20 0.32
CA14 Q9ULX7 1/20 0.32
SMO Q99835 1/20 0.32
TLR7 Q9NYK1 2/20 0.32
ABCG2 Q9UNQ0 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8566860 0.89 CA12 (0.34) DHFRKDM4EALDH1A1GLAGAA
SCHEMBL8572863 0.86 DHFR (0.37) SLC2A1DHFRALDH1A1MAPTHPGD
SCHEMBL27381948 0.79 ALDH1A1 (0.37) ALDH1A1
SCHEMBL8564223 0.75 TLR7 (0.37) SLC2A1DHFRKDM4EALDH1A1GLA
SCHEMBL8564228 0.75 TLR7 (0.37) SLC2A1DHFRKDM4EALDH1A1GLA
SCHEMBL8571595 0.73 TLR7 (0.38) SLC2A1DHFRKDM4EALDH1A1GLA
SCHEMBL8563771 0.72 TLR7 (0.45) CA12CA1CA2CA9CA14
SCHEMBL8564661 0.69 DHFR (0.39) DHFRALDH1A1MAPTHPGDTLR7
SCHEMBL6367420 0.67 TSHR (0.47) ALDH1A1MAPTCA12CA1CA2
SCHEMBL3643386 0.65 CA12 (0.48) KDM4EMAPTHPGDHIF1ATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530579-B1 Condensed pyrimidine derivatives antitumor agents EISAI CO LTD (JP) 1998-11-11 EP disclosed
US-5554615-A ANTITUMOR EISAI CO., LTD. (JP) 1996-09-10 US disclosed
EP-0530579-A1 Condensed pyrimidine derivatives antitumor agents Eisai Co., Ltd. (JP) 1993-03-10 EP disclosed