SCHEMBL8564673

SCHEMBL8564673

CC(C)(C)OC(=O)c1ccc(CCCn2ccc3nc(N)nc(N)c32)s1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATIC P31939 3/20 0.43
SHMT1 P34896 3/20 0.43
SHMT2 P34897 3/20 0.43
GART P22102 2/20 0.41
TLR7 Q9NYK1 8/20 0.37
DHFR P00374 2/20 0.34
SIRT2 Q8IXJ6 1/20 0.31
SIRT1 Q96EB6 1/20 0.31
SIRT3 Q9NTG7 1/20 0.31
HPGD P15428 3/20 0.30
KDM4E B2RXH2 2/20 0.30
ALDH1A1 P00352 2/20 0.30
GLA P06280 2/20 0.30
GAA P10253 2/20 0.30
MAPT P10636 2/20 0.30
HIF1A Q16665 2/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
THRB P10828 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8563771 0.81 TLR7 (0.45) ATICSHMT1SHMT2GARTTLR7
SCHEMBL8569300 0.75 ATIC (0.33) ATICSHMT1SHMT2GARTHPGD
SCHEMBL8564137 0.75 ATIC (0.75) ATICSHMT1SHMT2GART
SCHEMBL8564142 0.75 ATIC (0.75) ATICSHMT1SHMT2GART
SCHEMBL9001785 0.73 TLR7 (0.44) ATICSHMT1SHMT2GARTTLR7
SCHEMBL5050275 0.71 HPGD (0.42) HPGDALDH1A1
SCHEMBL9439883 0.71 FOLR1 (0.44) GART
SCHEMBL8571595 0.71 TLR7 (0.38) TLR7DHFRHPGDKDM4EALDH1A1
SCHEMBL9439499 0.70 DHFR (0.46) GARTDHFRSIRT2SIRT1SIRT3
SCHEMBL8570678 0.70 ATIC (0.38) ATICSHMT1SHMT2GARTTLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530579-B1 Condensed pyrimidine derivatives antitumor agents EISAI CO LTD (JP) 1998-11-11 EP disclosed
US-5554615-A ANTITUMOR EISAI CO., LTD. (JP) 1996-09-10 US disclosed
EP-0530579-A1 Condensed pyrimidine derivatives antitumor agents Eisai Co., Ltd. (JP) 1993-03-10 EP disclosed