SCHEMBL8564735

SCHEMBL8564735

CS(=O)(=O)Nc1cc[c]c(-c2ccc(S(N)(=O)=O)cc2)c1

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CA2 P00918 11/20 0.57
CA1 P00915 9/20 0.57
CA12 O43570 8/20 0.57
CA9 Q16790 7/20 0.57
MAPK8 P45983 1/20 0.43
MAPK10 P53779 1/20 0.43
CDK1 P06493 1/20 0.43
CDK2 P24941 1/20 0.43
KIF11 P52732 1/20 0.39
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CA14 Q9ULX7 2/20 0.38
CA4 P22748 1/20 0.38
CA6 P23280 1/20 0.38
CA5A P35218 1/20 0.38
CA7 P43166 1/20 0.38
CA5B Q9Y2D0 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9555262 0.75 CA1 (0.49) CA2CA1CA12CA9KIF11
SCHEMBL6401783 0.74 CA2 (1.00) CA2CA1CA12CA9MAPK8
SCHEMBL29899154 0.72 CA2 (0.63) CA2CA1CA12CA9ALDH1A1
SCHEMBL1765247 0.72 CA2 (0.63) CA2CA1CA12CA9ALDH1A1
SCHEMBL197213 0.70 ALDH1A1 (0.46) CA2CA1CA12CA9KIF11
SCHEMBL8594103 0.68 CA2 (0.57) CA2CA1CA12CA9CA14
SCHEMBL2896327 0.68 ALDH1A1 (0.45) CA2CA1CA12CA9KIF11
SCHEMBL1098358 0.68 ALDH1A1 (0.49) CA2CA1CA12CA9ALDH1A1
SCHEMBL314338 0.68 KIF11 (0.46) CA2CA1CA12CA9KIF11
SCHEMBL6608198 0.68 KEAP1 (0.53) CA2CA1CA12CA9KIF11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0431943-B1 Spiro(pyran)piperidine derivatives MERCK & CO INC (US) 1998-07-15 EP claimed
EP-0431943-B1 Spiro(pyran)piperidine derivatives MERCK & CO INC (US) 1998-07-15 EP disclosed
US-5633247-A ANTIARRTHYMIA AGENT MERCK & CO., INC. (US) 1997-05-27 US disclosed
US-5206240-A Antiarrhythmia agents MERCK & CO., INC. (US) 1993-04-27 US disclosed
EP-0431943-A2 Nitrogen-containing spirocycles MERCK & CO. INC. (US) 1991-06-12 EP disclosed