SCHEMBL8564661

SCHEMBL8564661

CC(Cc1ccc(C(=O)O)cc1)C(C)n1ccc2nc(N)nc(N)c21

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DHFR P00374 3/20 0.39
ANPEP P15144 1/20 0.39
ENPEP Q07075 1/20 0.39
TLR7 Q9NYK1 2/20 0.37
TLR8 Q9NR97 1/20 0.37
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
KMT2A Q03164 1/20 0.36
ATM Q13315 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
HSD17B10 Q99714 1/20 0.36
MBOAT4 Q96T53 1/20 0.34
ACACB O00763 1/20 0.33
FOLH1 Q04609 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8572863 0.82 DHFR (0.37) DHFRANPEPTLR7TLR8POLB
SCHEMBL8563902 0.71 TLR7 (0.50) DHFRTLR7POLBMAPTKMT2A
SCHEMBL8564668 0.70 ATIC (0.48) TLR7MAPTKMT2AALDH1A1
SCHEMBL8570466 0.69 DHFR (0.39) DHFRANPEPTLR7POLBMAPT
SCHEMBL8564762 0.69 SLC2A1 (0.34) DHFRTLR7MAPTKMT2AALDH1A1
SCHEMBL8564667 0.67 DHFR (0.38) DHFRTLR7POLBMAPTKMT2A
SCHEMBL251733 0.63 ANPEP (0.62) ANPEPENPEPALDH1A1
SCHEMBL2439514 0.63 ANPEP (0.62) ANPEPENPEPALDH1A1
SCHEMBL5183224 0.63 ANPEP (0.62) ANPEPENPEPALDH1A1
SCHEMBL452233 0.62 PTGS1 (0.60) ANPEPENPEPKMT2AALDH1A1ACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530579-B1 Condensed pyrimidine derivatives antitumor agents EISAI CO LTD (JP) 1998-11-11 EP disclosed
US-5554615-A ANTITUMOR EISAI CO., LTD. (JP) 1996-09-10 US disclosed
EP-0530579-A1 Condensed pyrimidine derivatives antitumor agents Eisai Co., Ltd. (JP) 1993-03-10 EP disclosed