SCHEMBL8564852

SCHEMBL8564852

c1ccc2c(c1)nc(N1CCCNCC1)c1cccn12

nearest known ligand 0.65

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 7/20 0.63
HTR3E A5X5Y0 6/20 0.63
HTR3B O95264 6/20 0.63
HTR3A P46098 6/20 0.63
HTR3D Q70Z44 6/20 0.63
HTR3C Q8WXA8 6/20 0.63
HTR1A P08908 6/20 0.63
HTR1D P28221 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8569563 0.87 HTR3E (0.75) HTR2CHTR3EHTR3BHTR3AHTR3D
SCHEMBL8569971 0.86 HTR3E (0.73) HTR2CHTR3EHTR3BHTR3AHTR3D
SCHEMBL17221919 0.85 HTR3E (0.69) HTR2CHTR3EHTR3BHTR3AHTR3D
SCHEMBL7301139 0.81 HTR1A (0.91) HTR2CHTR3EHTR3BHTR3AHTR3D
SCHEMBL8562640 0.79 HTR2C (0.69) HTR2CHTR3EHTR3BHTR3AHTR3D
SCHEMBL8564626 0.79 HTR3E (0.75) HTR2CHTR3EHTR3BHTR3AHTR3D
SCHEMBL2532527 0.79 HTR3E (0.66) HTR2CHTR3EHTR3BHTR3AHTR3D
SCHEMBL8564875 0.77 HTR3E (1.00) HTR2CHTR3EHTR3BHTR3AHTR3D
SCHEMBL8567791 0.77 HTR3E (0.74) HTR2CHTR3EHTR3BHTR3AHTR3D
SCHEMBL8571231 0.77 HTR3E (0.69) HTR2CHTR3EHTR3BHTR3AHTR3D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0623620-B1 5-HT3 Pyrrolopyrazine derivatives ADIR (FR) 1998-09-09 EP disclosed
US-5599812-A ANTISEROTONINE AGENTS ADIR ET COMPAGNIE (FR) 1997-02-04 US disclosed
EP-0623620-A1 5-HT3 Pyrrolopyrazine derivatives ADIR ET COMPAGNIE (FR) 1994-11-09 EP disclosed