SCHEMBL7415517

SCHEMBL7415517

O=C(N1CCc2ccc(-n3ccn(C4CCN(Cc5ccccc5)CC4)c3=O)cc2CC1)C(F)(F)F

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 3/20 0.43
DRD4 P21917 3/20 0.43
DRD3 P35462 3/20 0.43
NPY2R P49146 1/20 0.41
ACHE P22303 4/20 0.40
CHRM4 P08173 3/20 0.39
CHRM2 P08172 2/20 0.39
KDM4E B2RXH2 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
KMT2A Q03164 1/20 0.38
CHRM5 P08912 1/20 0.38
CHRM1 P11229 1/20 0.38
CHRM3 P20309 1/20 0.38
CXCR3 P49682 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7424664 0.85 DRD2 (0.43) DRD2DRD4DRD3LMNA
SCHEMBL7418940 0.84 ESR1 (0.42)
SCHEMBL8562233 0.78 ESR1 (0.39)
SCHEMBL8562237 0.78 ESR1 (0.39)
SCHEMBL8564898 0.77 ESR1 (0.39)
SCHEMBL8564893 0.77 ESR1 (0.39)
SCHEMBL3307108 0.72 ACHE (0.62) ACHECHRM4KDM4EALDH1A1LMNA
SCHEMBL7848854 0.71 HDAC3 (0.57) ACHEALDH1A1LMNAKMT2A
SCHEMBL7848948 0.70 CCR3 (0.54) DRD2DRD4DRD3ALDH1A1LMNA
SCHEMBL7478435 0.69 F10 (0.42) DRD4ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0777667-A1 CYCLIC BENZAZEPINE UREA DERIVATIVES WITH AGGREGATION-INHIBITING EFFECT Dr. Karl Thomae GmbH (DE) 1997-06-11 EP disclosed
WO-1996005194-A1 CYCLIC BENZAZEPINE UREA DERIVATIVES WITH AGGREGATION-INHIBITING EFFECT DR. KARL THOMAE GMBH (DE) 1996-02-22 WO disclosed