SCHEMBL8565728

SCHEMBL8565728

CC(C)(C)OC(=O)c1ccccc1C=S

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 1/20 0.39
ADRA1B P35368 1/20 0.39
HTT P42858 2/20 0.36
MEN1 O00255 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
KMT2A Q03164 1/20 0.36
TSHR P16473 3/20 0.36
ALDH1A1 P00352 2/20 0.36
HSD17B10 Q99714 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
GRM6 O15303 1/20 0.35
BACE1 P56817 1/20 0.35
LMNA P02545 3/20 0.34
ELANE P08246 1/20 0.34
BCHE P06276 1/20 0.34
GABRP O00591 1/20 0.34
GABRD O14764 1/20 0.34
GABRA1 P14867 1/20 0.34
GABRB1 P18505 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL97166 0.84 MEN1 (0.41) ADRA1AADRA1BHTTMEN1NPC1
SCHEMBL347774 0.83 CYP3A4 (0.40) ADRA1AADRA1BHTTMEN1NPC1
SCHEMBL30111657 0.81 TSHR (0.50) ADRA1AADRA1BHTTMEN1NPC1
SCHEMBL109178 0.81 TSHR (0.50) ADRA1AADRA1BHTTMEN1NPC1
Hydrogen Peroxide SCHEMBL29048859 0.79 TSHR (0.48) ADRA1AADRA1BHTTMEN1NPC1
SCHEMBL5074597 0.77 CYP3A4 (0.35) HTTNPC1TSHRALDH1A1HSD17B10
SCHEMBL20797216 0.76 PDK1 (0.37) ADRA1AADRA1BMEN1RAB9AKMT2A
SCHEMBL10514026 0.74 TSHR (0.44) ADRA1AADRA1BHTTMEN1NPC1
SCHEMBL39310 0.74 LMNA (0.62) ADRA1AADRA1BHTTKMT2ATSHR
SCHEMBL722115 0.74 ALDH1A1 (0.56) TSHRALDH1A1HSD17B10TDP1GRM6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530579-B1 Condensed pyrimidine derivatives antitumor agents EISAI CO LTD (JP) 1998-11-11 EP disclosed
US-5688800-A ANTITUMOR AGENTS EISAI CO., LTD. (JP) 1997-11-18 US disclosed
US-5554615-A ANTITUMOR EISAI CO., LTD. (JP) 1996-09-10 US disclosed
EP-0530579-A1 Condensed pyrimidine derivatives antitumor agents Eisai Co., Ltd. (JP) 1993-03-10 EP disclosed