SCHEMBL8565869

SCHEMBL8565869

CN1CCN(c2ncnc(Cl)c2Sc2ccc(Cl)cc2)CC1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.67
DRD2 P14416 3/20 0.67
DRD4 P21917 3/20 0.67
NPC1 O15118 1/20 0.48
GAA P10253 1/20 0.48
RAB9A P51151 1/20 0.48
HRH4 Q9H3N8 6/20 0.47
CNR1 P21554 2/20 0.42
KCNH2 Q12809 2/20 0.42
HTT P42858 1/20 0.42
KMT2A Q03164 1/20 0.41
HTR3B O95264 1/20 0.40
HTR3A P46098 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
HSD17B10 Q99714 1/20 0.40
MAPK13 O15264 1/20 0.40
MAPK12 P53778 1/20 0.40
MAPK11 Q15759 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8569210 0.89 HTR1A (0.62) HTR1ADRD2DRD4HRH4HTT
SCHEMBL8566405 0.79 CYP1A2 (0.50) HTR1ADRD2DRD4HRH4CNR1
SCHEMBL8564570 0.77 HTR1A (0.82) HTR1ADRD2DRD4
SCHEMBL8569140 0.75 L3MBTL1 (0.46) HTR1ADRD2DRD4HTTKMT2A
SCHEMBL30828999 0.74 HTT (0.56) NPC1GAARAB9AHRH4HTT
SCHEMBL26647139 0.74 HTT (0.56) NPC1GAARAB9AHRH4HTT
SCHEMBL28638711 0.68 CYP1A2 (0.67) NPC1GAARAB9AHRH4HTT
SCHEMBL8565639 0.67 HTR1A (1.00) HTR1ADRD2DRD4HRH4
SCHEMBL8567179 0.67 HTR1A (0.67) HTR1ADRD2DRD4HRH4HTR3B
SCHEMBL4366557 0.67 CYP3A4 (0.70) HRH4HTTKMT2ACYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0826674-A1 NOVEL PYRIMIDINE DERIVATIVES EFFICACIOUS AS PSYCHOTROPIC DRUG AND PROCESS FOR THE PRODUCTION THEREOF SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1998-03-04 EP disclosed