SCHEMBL9001791

SCHEMBL9001791

Nc1nc(O)c2c(n1)CCC2CCc1ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)o1

nearest known ligand 0.66

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ATIC P31939 2/20 0.46
FOLR2 P14207 1/20 0.46
FOLR1 P15328 1/20 0.46
DHFR P00374 6/20 0.43
MTR Q99707 1/20 0.43
TYMS P04818 1/20 0.40
GART P22102 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9001930 0.95 ATIC (0.48) ATICFOLR2FOLR1DHFRMTR
SCHEMBL8568731 0.92 DHFR (0.47) ATICFOLR2FOLR1DHFRMTR
SCHEMBL8565987 0.88 FOLR2 (0.49) ATICFOLR2FOLR1DHFRMTR
SCHEMBL9001801 0.87 DHFR (0.53) ATICDHFRMTRTYMSGART
SCHEMBL9001799 0.84 DHFR (0.54) ATICDHFRMTRTYMSGART
SCHEMBL9001752 0.84 GART (0.53) ATICFOLR2FOLR1GART
SCHEMBL9001769 0.81 FOLR1 (0.49) ATICFOLR2FOLR1GART
SCHEMBL8571475 0.79 DHFR (0.57) DHFRMTRGART
SCHEMBL9387643 0.78 GART (0.59) ATICFOLR2FOLR1DHFRGART
SCHEMBL9387634 0.78 GART (0.59) ATICFOLR2FOLR1DHFRGART

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5554615-A ANTITUMOR EISAI CO., LTD. (JP) 1996-09-10 US disclosed
EP-0530579-A1 Condensed pyrimidine derivatives antitumor agents Eisai Co., Ltd. (JP) 1993-03-10 EP disclosed