SCHEMBL8566680

SCHEMBL8566680

COC(=O)Cc1nsc(NC(=O)c2ccccc2)n1

nearest known ligand 0.76

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.60
NPC1 O15118 3/20 0.57
ADORA3 P0DMS8 7/20 0.57
ALDH1A1 P00352 5/20 0.53
KDM4E B2RXH2 2/20 0.51
RXFP1 Q9HBX9 1/20 0.51
HTT P42858 1/20 0.51
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
HSD17B10 Q99714 1/20 0.50
MAPT P10636 2/20 0.47
LMNA P02545 2/20 0.47
USP2 O75604 1/20 0.47
HPGD P15428 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
RAB9A P51151 2/20 0.47
PKM P14618 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8565133 0.89 ALDH1A1 (0.61) NPSR1NPC1ADORA3ALDH1A1KDM4E
SCHEMBL8570794 0.86 ADORA3 (0.62) NPC1ADORA3ALDH1A1KDM4ERXFP1
SCHEMBL8565123 0.82 ALDH1A1 (0.49) NPC1ALDH1A1KDM4EHTTMEN1
SCHEMBL8570956 0.81 ADORA3 (0.53) NPSR1NPC1ADORA3ALDH1A1KDM4E
SCHEMBL8573320 0.79 NPC1 (0.44) NPC1ALDH1A1KDM4EHTTMEN1
SCHEMBL8570862 0.78 ADORA3 (0.59) NPC1ADORA3ALDH1A1KDM4ERXFP1
SCHEMBL30911334 0.77 ADORA3 (0.61) NPC1ADORA3KDM4ERXFP1KMT2A
SCHEMBL8575278 0.77 ADORA3 (0.51) NPC1ADORA3ALDH1A1KDM4ERXFP1
SCHEMBL1377141 0.76 ADORA3 (0.68) NPC1ADORA3RXFP1MEN1KMT2A
SCHEMBL8568489 0.75 NPC1 (0.48) NPC1ALDH1A1KDM4EHTTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5705650-A Process for preparing 1,2,4-thiadiazole derivatives KATAYAMA SEIYAKUSYO CO., LTD. (JP) 1998-01-06 US disclosed
US-5585494-A Process for preparing 1,2,4-thiadiazole derivatives KATAYAMA SEIYAKUSYO CO. LTD. (JP) 1996-12-17 US disclosed
EP-0536900-A2 Process for preparing 1,2,4-Thiadiazole Derivatives KATAYAMA SEIYAKUSYO CO. Ltd. (JP) 1993-04-14 EP disclosed