SCHEMBL8568489

SCHEMBL8568489

COC(=O)Cc1nsc(NC(=O)C(C)(C)C)n1

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 7/20 0.48
SMN1; SMN2 Q16637 6/20 0.48
RAB9A P51151 6/20 0.48
LMNA P02545 2/20 0.48
TP53 P04637 1/20 0.48
POLB P06746 1/20 0.48
NFKB1 P19838 1/20 0.48
NFKB2 Q00653 1/20 0.48
RELA Q04206 1/20 0.48
ALDH1A1 P00352 7/20 0.42
MAPT P10636 2/20 0.42
HPGD P15428 1/20 0.42
KDM4E B2RXH2 2/20 0.40
HTT P42858 1/20 0.40
MEN1 O00255 1/20 0.40
CYP1A2 P05177 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8573320 0.83 NPC1 (0.44) NPC1SMN1; SMN2RAB9ALMNAALDH1A1
SCHEMBL9564508 0.79 SMN1; SMN2 (0.48) NPC1SMN1; SMN2RAB9ALMNAALDH1A1
SCHEMBL6761097 0.78 ALDH1A1 (0.43) NPC1SMN1; SMN2RAB9ALMNAALDH1A1
SCHEMBL8566680 0.75 NPSR1 (0.60) NPC1SMN1; SMN2RAB9ALMNAALDH1A1
SCHEMBL8572394 0.73 NPC1 (0.41) NPC1SMN1; SMN2RAB9ALMNAALDH1A1
SCHEMBL8565123 0.73 ALDH1A1 (0.49) NPC1SMN1; SMN2RAB9ALMNAPOLB
SCHEMBL24491025 0.73 RAB9A (0.56) NPC1SMN1; SMN2RAB9ALMNATP53
SCHEMBL16425168 0.73 HSD17B10 (0.39) NPC1SMN1; SMN2RAB9ALMNAALDH1A1
SCHEMBL8568524 0.72 TSHR (0.43) NPC1SMN1; SMN2RAB9ALMNAPOLB
SCHEMBL10840353 0.71 SMN1; SMN2 (0.43) SMN1; SMN2LMNAPOLBALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5705650-A Process for preparing 1,2,4-thiadiazole derivatives KATAYAMA SEIYAKUSYO CO., LTD. (JP) 1998-01-06 US disclosed
US-5585494-A Process for preparing 1,2,4-thiadiazole derivatives KATAYAMA SEIYAKUSYO CO. LTD. (JP) 1996-12-17 US disclosed
EP-0536900-A2 Process for preparing 1,2,4-Thiadiazole Derivatives KATAYAMA SEIYAKUSYO CO. Ltd. (JP) 1993-04-14 EP disclosed