SCHEMBL8568940

SCHEMBL8568940

COC(=O)C(N)c1ccccc1N

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.47
HSD17B10 Q99714 3/20 0.47
CFTR P13569 1/20 0.47
KMT2A Q03164 2/20 0.44
ADRA2B P18089 1/20 0.41
PTGS1 P23219 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
HDAC3 O15379 1/20 0.37
HDAC4 P56524 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC7 Q8WUI4 1/20 0.37
HDAC2 Q92769 1/20 0.37
HDAC10 Q969S8 1/20 0.37
HDAC11 Q96DB2 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
HDAC9 Q9UKV0 1/20 0.37
HDAC5 Q9UQL6 1/20 0.37
TSHR P16473 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9664845 0.88 KMT2A (0.50) ALDH1A1HSD17B10CFTRKMT2APTGS1
SCHEMBL28996258 0.83 ALDH1A1 (0.56) ALDH1A1HSD17B10CFTRKMT2AADRA2B
SCHEMBL7976422 0.81 CA1 (0.47) ALDH1A1KMT2AADRA2BPTGS1TDP1
SCHEMBL11330367 0.81 ALDH1A1 (0.47) ALDH1A1HSD17B10CFTRKMT2AADRA2B
SCHEMBL2635055 0.81 ALDH1A1 (0.47) ALDH1A1HSD17B10CFTRKMT2APTGS1
SCHEMBL7203924 0.81 AAK1 (0.39) ALDH1A1HSD17B10CFTRKMT2AADRA2B
SCHEMBL15670602 0.80 KMT2A (0.47) ALDH1A1KMT2APOLB
SCHEMBL1159853 0.80 CASP1 (0.44) ALDH1A1KMT2A
SCHEMBL21296572 0.80 CYP2C19 (0.44) ALDH1A1KMT2APOLBCYP3A4
SCHEMBL15670601 0.80 KMT2A (0.47) ALDH1A1KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5719141-A HYPOTENSIVE AGENTS NOVARTIS CORPORATION (US) 1998-02-17 US disclosed
EP-0702004-A2 2,9-diamino- and 2-amino-8-carbamoyl-4-hydroxy-alkanoic acid amid derivatives CIBA-GEIGY AG (CH) 1996-03-20 EP disclosed