SCHEMBL8569451

SCHEMBL8569451

COc1ccc(Oc2ccccc2)cc1C(=O)N(C)OC

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.49
POLB P06746 1/20 0.49
TTR P02766 1/20 0.47
F2 P00734 1/20 0.45
F10 P00742 1/20 0.45
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
PLA2G2A P14555 1/20 0.44
BACE1 P56817 1/20 0.44
MAPT P10636 1/20 0.43
HTT P42858 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
HSD11B1 P28845 1/20 0.43
ALDH1A1 P00352 1/20 0.43
TSHR P16473 1/20 0.42
LTA4H P09960 1/20 0.42
ALOX5 P09917 1/20 0.42
PTGS1 P23219 1/20 0.42
PTGS2 P35354 1/20 0.42
RAB9A P51151 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4833864 0.85 MAPT (0.58) KDM4EPOLBMEN1KMT2AMAPT
SCHEMBL8572013 0.82 KDM4E (0.69) KDM4EPOLBTTRPLA2G2AMAPT
SCHEMBL8573443 0.80 NR1H4 (0.49) KDM4EPOLBMEN1KMT2ATSHR
SCHEMBL31605270 0.78 ALDH1A1 (0.63) KDM4EPOLBMEN1KMT2AMAPT
SCHEMBL11474623 0.78 MAPT (0.56) MEN1KMT2AMAPTHTTNPSR1
SCHEMBL19533698 0.77 SMN1; SMN2 (0.59) KDM4EPOLBMEN1KMT2AALDH1A1
SCHEMBL8577030 0.77 ACHE (0.47) KDM4EPOLBMEN1KMT2AMAPT
SCHEMBL307126 0.77 CTSD (0.51) HTTRAB9A
SCHEMBL8570550 0.75 MEN1 (0.53) KDM4EPOLBTTRMEN1KMT2A
SCHEMBL5623892 0.75 TSHR (0.57) POLBMEN1KMT2AMAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5739336-A SELECTIVE 5-HYDROXYTRYPTAMINE-2C RECEPTOR ANTAGONISTS SYNTEX (U.S.A.) INC. (US) 1998-04-14 US disclosed
WO-1997000872-A1 1,3,8-TRIAZA- AND 3,8-DIAZA-1-OXASPIRO(4,5)DECANE DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 1997-01-09 WO disclosed