SCHEMBL8569656

SCHEMBL8569656

CCCCOC(=O)N[C@H](CC#N)C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CTSS P25774 4/20 0.43
CTSL P07711 1/20 0.43
CTSK P43235 3/20 0.43
EPHX1 P07099 1/20 0.40
ACHE P22303 7/20 0.39
ITGB3 P05106 2/20 0.39
ITGA2B P08514 2/20 0.39
ALDH1A1 P00352 1/20 0.38
NPC1 O15118 1/20 0.38
HPGD P15428 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8564079 0.91 CTSS (0.38) CTSSCTSLCTSKITGB3ITGA2B
SCHEMBL8561162 0.88 CTSS (0.41) CTSSCTSLCTSKEPHX1ACHE
SCHEMBL16119729 0.85 CTSS (0.47) CTSSCTSLCTSKEPHX1ACHE
SCHEMBL1895877 0.85 CYP1A2 (0.40) EPHX1ACHEITGB3ITGA2BALDH1A1
SCHEMBL3645507 0.84 MMP3 (0.40) EPHX1ACHEITGB3ITGA2BALDH1A1
SCHEMBL480292 0.82 EPHX1 (0.46) CTSKEPHX1ACHEITGB3ITGA2B
SCHEMBL284168 0.82 EPHX1 (0.46) CTSKEPHX1ACHEITGB3ITGA2B
Water SCHEMBL27304038 0.81 PLA2G2A (0.54) ALDH1A1
SCHEMBL21359118 0.81 HRH3 (0.42) EPHX1ACHENPC1HPGDRAB9A
Water SCHEMBL4794958 0.81 PLA2G2A (0.54) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0821675-A1 NOVEL HYDROXAMIC ACID AND AMINO-CARBOXYLATE COMPOUNDS AS METALLOPROTEASE AND TNF INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1998-02-04 EP disclosed
US-5703092-A TREATING ARTHRITIS, OTHER INFLAMMATORY DISEASES MEDIATED BY MATRIX METALLOPROTEINASE AND/OR TUMOR NECROSIS FACTOR THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1997-12-30 US disclosed
WO-1996033176-A1 NOVEL HYDROXAMIC ACID AND AMINO-CARBOXYLATE COMPOUNDS AS METALLOPROTEASE AND TNF INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-10-24 WO disclosed