SCHEMBL8570466

SCHEMBL8570466

CCC(Cn1ccc2nc(N)nc(N)c21)c1ccc(C(=O)O)cc1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DHFR P00374 8/20 0.39
TLR7 Q9NYK1 1/20 0.37
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
KMT2A Q03164 1/20 0.36
ATM Q13315 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
HSD17B10 Q99714 1/20 0.36
ANPEP P15144 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8564667 0.89 DHFR (0.38) DHFRTLR7POLBMAPTKMT2A
SCHEMBL8564196 0.82 DHFR (0.58) DHFR
SCHEMBL8572863 0.78 DHFR (0.37) DHFRTLR7POLBMAPTKMT2A
SCHEMBL8561990 0.74 DHFR (0.57) DHFR
SCHEMBL8563902 0.74 TLR7 (0.50) DHFRTLR7POLBMAPTKMT2A
SCHEMBL19910225 0.72 SLC2A1 (0.58) DHFRTLR7POLB
SCHEMBL8564668 0.72 ATIC (0.48) TLR7MAPTKMT2AALDH1A1
SCHEMBL22730044 0.70 CDK1 (0.44) DHFRTLR7
SCHEMBL8570681 0.69 ATIC (0.49) DHFR
SCHEMBL8567007 0.69 DHFR (0.47) DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530579-B1 Condensed pyrimidine derivatives antitumor agents EISAI CO LTD (JP) 1998-11-11 EP disclosed
US-5554615-A ANTITUMOR EISAI CO., LTD. (JP) 1996-09-10 US disclosed
EP-0530579-A1 Condensed pyrimidine derivatives antitumor agents Eisai Co., Ltd. (JP) 1993-03-10 EP disclosed