SCHEMBL8563902

SCHEMBL8563902

Nc1nc(N)c2c(ccn2CCCc2ccc(C(=O)O)cc2)n1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TLR7 Q9NYK1 1/20 0.50
ATIC P31939 3/20 0.46
SHMT1 P34896 3/20 0.46
SHMT2 P34897 3/20 0.46
TBXAS1 P24557 2/20 0.46
GART P22102 2/20 0.44
EP300 Q09472 6/20 0.43
DHFR P00374 1/20 0.39
POLB P06746 1/20 0.39
MAPT P10636 1/20 0.39
KMT2A Q03164 1/20 0.39
ATM Q13315 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
RARB P10826 1/20 0.38
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
HSD17B10 Q99714 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8564668 0.95 ATIC (0.48) TLR7ATICSHMT1SHMT2TBXAS1
SCHEMBL8563771 0.84 TLR7 (0.45) TLR7ATICSHMT1SHMT2GART
SCHEMBL8563883 0.80 ATIC (0.74) ATICSHMT1SHMT2GARTDHFR
SCHEMBL8563875 0.80 ATIC (0.74) ATICSHMT1SHMT2GARTDHFR
SCHEMBL8564667 0.77 DHFR (0.38) TLR7DHFRPOLBMAPTKMT2A
SCHEMBL9001785 0.76 TLR7 (0.44) TLR7ATICSHMT1SHMT2TBXAS1
SCHEMBL8570466 0.74 DHFR (0.39) TLR7DHFRPOLBMAPTKMT2A
SCHEMBL9001870 0.74 ATIC (0.73) ATICSHMT1SHMT2GARTDHFR
SCHEMBL8567736 0.73 ATIC (0.66) ATICSHMT1SHMT2GARTDHFR
SCHEMBL8567743 0.73 ATIC (0.66) ATICSHMT1SHMT2GARTDHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0530579-B1 Condensed pyrimidine derivatives antitumor agents EISAI CO LTD (JP) 1998-11-11 EP disclosed
US-5554615-A ANTITUMOR EISAI CO., LTD. (JP) 1996-09-10 US disclosed
EP-0530579-A1 Condensed pyrimidine derivatives antitumor agents Eisai Co., Ltd. (JP) 1993-03-10 EP disclosed