SCHEMBL8570815

SCHEMBL8570815

CC[C@H]1CSc2ccccc2[C@@H](c2ccccc2)C1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 7/20 0.40
ADRA1A P35348 4/20 0.38
HTR2A P28223 2/20 0.37
HTR2C P28335 2/20 0.37
HTR2B P41595 2/20 0.37
HRH3 Q9Y5N1 2/20 0.37
HTR1A P08908 2/20 0.37
ADRA1D P25100 2/20 0.37
ADRA1B P35368 2/20 0.37
MTNR1A P48039 1/20 0.36
MTNR1B P49286 1/20 0.36
MEN1 O00255 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
ALOX15 P16050 1/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36
CYP2C19 P33261 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9565765 0.78 MEN1 (0.44) SIGMAR1MEN1CYP3A4KMT2A
SCHEMBL12463825 0.70 SLC6A2 (0.38) MEN1KMT2A
SCHEMBL29100535 0.68 USP2 (0.46) MEN1KMT2A
SCHEMBL6221558 0.68 SLC10A2 (0.40) SIGMAR1HTR2AHTR2CHTR2BHRH3
SCHEMBL6221549 0.68 SLC10A2 (0.40) SIGMAR1HTR2AHTR2CHTR2BHRH3
SCHEMBL7419856 0.66 KMT2A (0.40) SIGMAR1MEN1KMT2A
SCHEMBL13843475 0.66 ALDH1A1 (0.42) HTR2BMEN1CYP1A2CYP3A4ALOX15
SCHEMBL1388099 0.66 SIGMAR1 (0.55) SIGMAR1HTR2AHTR2CHTR2BHRH3
SCHEMBL11548867 0.65 SIGMAR1 (0.44) SIGMAR1HTR2AHTR2CHTR2BHRH3
SCHEMBL27173470 0.64 LMNA (0.41) SIGMAR1MEN1TSHRKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997033882-A9 NOVEL BENZOTHIEPINES HAVING ACTIVITY AS INHIBITORS OF ILEAL BILE ACID TRANSPORT AND TAUROCHOLATE UPTAKE 1998-02-26 WO disclosed