SCHEMBL8577149

SCHEMBL8577149

NCC1CNCCC1Nc1ccc(F)c(Cl)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.40
MAPKAPK2 P49137 4/20 0.38
KMT2A Q03164 3/20 0.38
CDK2 P24941 3/20 0.38
ALDH1A1 P00352 3/20 0.38
MEN1 O00255 2/20 0.38
SLC6A2 P23975 3/20 0.38
NR1I2 O75469 1/20 0.38
AHR P35869 1/20 0.38
SLC6A4 P31645 2/20 0.36
SLC6A3 Q01959 2/20 0.36
RPS6KB1 P23443 2/20 0.36
AKT1 P31749 2/20 0.36
MAPT P10636 1/20 0.35
HTT P42858 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
SOS1 Q07889 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
ABL1 P00519 1/20 0.35
RECQL P46063 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8572372 0.83 KMT2A (0.40) TRPA1MAPKAPK2KMT2ACDK2ALDH1A1
SCHEMBL8572427 0.76 KMT2A (0.44) TRPA1KMT2AALDH1A1MEN1NR1I2
Hydrochloric Acid SCHEMBL5178097 0.71 SLC6A2 (0.41) SLC6A2SLC6A4SLC6A3
SCHEMBL8577356 0.70 ALDH1A1 (0.40) TRPA1MAPKAPK2KMT2ACDK2ALDH1A1
SCHEMBL27262054 0.69 SLC6A2 (0.45) MAPKAPK2CDK2SLC6A2
SCHEMBL9008342 0.68 KMT2A (0.59) TRPA1MAPKAPK2KMT2ACDK2ALDH1A1
SCHEMBL31453688 0.68 KMT2A (0.59) TRPA1MAPKAPK2KMT2ACDK2ALDH1A1
SCHEMBL29458485 0.68 MALT1 (0.58) KMT2AALDH1A1MEN1NR1I2AHR
SCHEMBL22644321 0.68 MALT1 (0.58) KMT2AALDH1A1MEN1NR1I2AHR
SCHEMBL8574181 0.68 MAPKAPK2 (0.44) TRPA1MAPKAPK2KMT2ACDK2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5821240-A ENZYME INHIBITORS, SIGNAL INHIBITORS FOR ANTIINFLAMMATORY AGENTS, ANTICARCINOGENIC AGENTS, ANTITUMOR AGENTS AND HORMONE INHIBITORS DR. KARL THOMAE GMBH (DE) 1998-10-13 US disclosed