SCHEMBL8577356

SCHEMBL8577356

NCC1CC(Nc2ccc(F)c(Cl)c2)CCN1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.40
KMT2A Q03164 4/20 0.40
MEN1 O00255 3/20 0.40
TRPA1 O75762 1/20 0.40
MAPKAPK2 P49137 2/20 0.38
NR1I2 O75469 1/20 0.38
AHR P35869 1/20 0.38
MAP3K8 P41279 1/20 0.36
MAPT P10636 1/20 0.35
HTT P42858 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
RAPGEF4 Q8WZA2 1/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
ABL1 P00519 1/20 0.35
RECQL P46063 1/20 0.35
RIN1 Q13671 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
KCNH2 Q12809 1/20 0.35
TSHR P16473 1/20 0.35
PLA2G1B P04054 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9008342 0.74 KMT2A (0.59) ALDH1A1KMT2AMEN1TRPA1MAPKAPK2
SCHEMBL31453688 0.74 KMT2A (0.59) ALDH1A1KMT2AMEN1TRPA1MAPKAPK2
SCHEMBL8574021 0.72 TRPA1 (0.40) ALDH1A1KMT2AMEN1TRPA1MAPKAPK2
SCHEMBL8574181 0.70 MAPKAPK2 (0.44) ALDH1A1KMT2AMEN1TRPA1MAPKAPK2
SCHEMBL8573402 0.70 KMT2A (0.43) ALDH1A1KMT2AMEN1TRPA1MAPKAPK2
SCHEMBL8577149 0.70 TRPA1 (0.40) ALDH1A1KMT2AMEN1TRPA1MAPKAPK2
SCHEMBL27598965 0.69 TRPA1 (0.46) ALDH1A1KMT2AMEN1TRPA1MAPKAPK2
SCHEMBL8572427 0.68 KMT2A (0.44) ALDH1A1KMT2AMEN1TRPA1NR1I2
SCHEMBL8575860 0.68 MAPKAPK2 (0.43) ALDH1A1KMT2AMEN1TRPA1MAPKAPK2
SCHEMBL8572544 0.68 KMT2A (0.46) ALDH1A1KMT2AMEN1TRPA1NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5821240-A ENZYME INHIBITORS, SIGNAL INHIBITORS FOR ANTIINFLAMMATORY AGENTS, ANTICARCINOGENIC AGENTS, ANTITUMOR AGENTS AND HORMONE INHIBITORS DR. KARL THOMAE GMBH (DE) 1998-10-13 US disclosed