SCHEMBL8577219

SCHEMBL8577219

CCOc1ccc(N)c(C(=O)c2ccc3c(c2)OCO3)c1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.48
LMNA P02545 1/20 0.48
TSHR P16473 1/20 0.48
MAPT P10636 5/20 0.47
RAB9A P51151 5/20 0.46
NPC1 O15118 3/20 0.46
SRD5A2 P31213 1/20 0.46
CTNNB1 P35222 1/20 0.46
WNT3A P56704 1/20 0.46
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
ALDH1A1 P00352 1/20 0.45
KDM4E B2RXH2 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5823399 0.86 CTNNB1 (0.57) SMN1; SMN2LMNAMAPTRAB9ANPC1
SCHEMBL22230088 0.84 MAPT (0.56) SMN1; SMN2LMNAMAPTRAB9ANPC1
SCHEMBL22230026 0.82 MAPT (0.55) SMN1; SMN2LMNAMAPTRAB9ANPC1
SCHEMBL3522633 0.78 MAPT (0.60) SMN1; SMN2LMNAMAPTRAB9ANPC1
SCHEMBL984344 0.76 MAOB (0.62) SMN1; SMN2LMNATSHRMAPTRAB9A
SCHEMBL8301109 0.74 RAB9A (0.61) SMN1; SMN2LMNAMAPTRAB9ANPC1
SCHEMBL21834006 0.73 ALDH1A1 (0.66) SMN1; SMN2LMNAMAPTRAB9ANPC1
SCHEMBL21833994 0.73 ALDH1A1 (0.56) SMN1; SMN2LMNAMAPTRAB9ANPC1
SCHEMBL8525053 0.72 RAB9A (0.48) SMN1; SMN2LMNAMAPTRAB9ANPC1
SCHEMBL28471046 0.72 MAPT (0.65) SMN1; SMN2LMNATSHRMAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5731321-A Endothelin receptor antagonists MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1998-03-24 US disclosed
EP-0757039-A1 Endothelin receptor antagonists MERCK PATENT GmbH (DE) 1997-02-05 EP disclosed