SCHEMBL8577922

SCHEMBL8577922

COC(=O)CCC1CN(c2ccc(C#N)c(F)c2)C(=O)N1c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 4/20 0.41
CHRM1 P11229 3/20 0.41
CHRM5 P08912 1/20 0.41
CHRM4 P08173 2/20 0.39
KDM1A O60341 8/20 0.36
DPP4 P27487 1/20 0.35
PREP P48147 1/20 0.35
DPP8 Q6V1X1 1/20 0.35
DPP9 Q86TI2 1/20 0.35
DPP7 Q9UHL4 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
ALDH1A1 P00352 1/20 0.35
HPGD P15428 1/20 0.35
TSHR P16473 1/20 0.35
USP14 P54578 1/20 0.35
PDE4B Q07343 1/20 0.34
PDE4D Q08499 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8577063 0.89 AR (0.43) AR
SCHEMBL8573438 0.84 CTSG (0.40) CHRM2CHRM4HDAC1HDAC6ALDH1A1
SCHEMBL8575471 0.84 PTGER4 (0.36) CHRM4ALDH1A1TSHR
Hydrochloric Acid SCHEMBL8571485 0.83 CTSG (0.39) CHRM2CHRM4HDAC1HDAC6ALDH1A1
Hydrochloric Acid SCHEMBL8573565 0.79 CTSG (0.39) ALDH1A1TSHR
SCHEMBL8575669 0.79 CTSG (0.39) CHRM2CHRM4ALDH1A1TSHR
SCHEMBL8571584 0.78 CTSG (0.39) HDAC1ALDH1A1HPGDTSHR
SCHEMBL8571508 0.77 HTR7 (0.37) HPGDTSHR
SCHEMBL8575092 0.77 CTSG (0.43) ALDH1A1TSHR
SCHEMBL8572736 0.77 OPRM1 (0.43) ALDH1A1HPGDAR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5852192-A Cyclic urea derivatives, pharmaceutical compositions containing these compounds and processes for preparing them DR. KARL THOMAE GMBH (DE) 1998-12-22 US disclosed