SCHEMBL8600706

SCHEMBL8600706

S=c1cc[nH]c2cc(Cc3ccccc3)ccc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FEN1 P39748 1/20 0.43
GPR17 Q13304 1/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
IDH1 O75874 1/20 0.40
CALM1 P0DP23 1/20 0.39
CYP2C9 P11712 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38
GSK3B P49841 1/20 0.38
GABRA1 P14867 2/20 0.36
GABRB2 P47870 2/20 0.36
ALDH1A1 P00352 1/20 0.36
HPGD P15428 1/20 0.36
PTGES O14684 1/20 0.35
HNF4A P41235 1/20 0.35
GABRB1 P18505 1/20 0.34
GABRA3 P34903 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8603411 0.78 RHEB (0.42) MEN1KMT2AALDH1A1
SCHEMBL7504545 0.76 BACE1 (0.48) MEN1KMT2AIDH1CALM1CYP2D6
SCHEMBL8600722 0.76 MAOA (0.43) MEN1KMT2ACYP3A4
SCHEMBL8602858 0.76 IMPDH2 (0.56) GABRA1ALDH1A1HPGDGABRA3
SCHEMBL8600219 0.75 MAOA (0.43) MEN1KMT2AALDH1A1
SCHEMBL8602871 0.75 NPC1 (0.53) FEN1GPR17MEN1KMT2AGSK3B
SCHEMBL8603563 0.74 PARP1 (0.39) MEN1KMT2ACYP3A4CYP2D6CYP2C19
SCHEMBL30030142 0.73 CYP17A1 (0.55) CYP2D6
SCHEMBL8604113 0.73 CYP17A1 (0.55) CYP2D6
SCHEMBL8603453 0.71 RELA (0.41) CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5773449-A BACTERICIDES FOR HELICOBACTER ZENYAKU KOGYO KABUSHIKI KAISHA (JP) 1998-06-30 US disclosed
EP-0786454-A1 THIOQUINOLONE DERIVATIVE ZENYAKU KOGYO KABUSHIKIKAISHA (JP) 1997-07-30 EP disclosed