SCHEMBL8600809

SCHEMBL8600809

COc1ccc2cc(C3(O)CCCC3)sc2c1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.44
CHRNA7 P36544 3/20 0.40
SIGMAR1 Q99720 3/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C19 P33261 1/20 0.38
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38
BCHE P06276 1/20 0.37
PDK1 Q15118 1/20 0.37
BACE1 P56817 1/20 0.36
NPC1 O15118 1/20 0.36
MAPT P10636 1/20 0.36
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8596068 0.99 CA2 (0.43) CA2CHRNA7SIGMAR1MAOAMAOB
SCHEMBL8600765 0.99 CA2 (0.43) CA2CHRNA7SIGMAR1MAOAMAOB
SCHEMBL4444185 0.99 CA2 (0.43) CA2CHRNA7SIGMAR1MAOAMAOB
SCHEMBL8599290 0.86 CHRNA7 (0.42) CA2CHRNA7CYP1A2CYP3A4CYP2C19
SCHEMBL8598275 0.85 CHRNA7 (0.39) CA2CHRNA7MAOAMAOBNPC1
SCHEMBL8598239 0.84 CA2 (0.39) CA2CHRNA7CYP1A2CYP3A4CYP2C19
SCHEMBL8626160 0.83 MAPT (0.43) CA2CHRNA7CYP1A2CYP3A4CYP2C19
SCHEMBL8597630 0.80 MAPT (0.45) CA2CHRNA7MAOAMAOBNPC1
SCHEMBL6311972 0.78 ALDH1A1 (0.46) CHRNA7BACE1MAPT
SCHEMBL1628516 0.73 CYP1A2 (0.46) CYP1A2BCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0641791-B1 NOVEL BENZOTHIOPHENE DERIVATIVE TEIKOKU HORMONE MFG CO LTD (JP) 1998-01-28 EP disclosed
US-5472962-A Antiestrogenic agents TEIKOKU HORMONE MFG. CO., LTD. (JP) 1995-12-05 US disclosed
EP-0641791-A1 NOVEL BENZOTHIOPHENE DERIVATIVE TEIKOKU HORMONE MFG. CO., LTD. (JP) 1995-03-08 EP disclosed