SCHEMBL8601267

SCHEMBL8601267

Cc1cn(Cc2ccc3c(c2)OCO3)c2cc(C3CCNC3=O)ccc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.49
PDE4B Q07343 1/20 0.49
PDE4C Q08493 1/20 0.49
PDE4D Q08499 1/20 0.49
SLC22A12 Q96S37 1/20 0.44
CHRNB2 P17787 1/20 0.41
CHRNA7 P36544 1/20 0.41
CHRNA4 P43681 1/20 0.41
CMA1 P23946 1/20 0.40
TSHR P16473 5/20 0.39
ALDH1A1 P00352 3/20 0.39
USP2 O75604 3/20 0.39
GAA P10253 1/20 0.39
MAPK1 P28482 1/20 0.39
PDE5A O76074 2/20 0.39
PDE1A P54750 2/20 0.38
PDE1B Q01064 2/20 0.38
PDE1C Q14123 2/20 0.38
POLB P06746 1/20 0.38
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8599642 0.84 PDE4A (0.44) PDE4APDE4BPDE4CPDE4DSLC22A12
SCHEMBL8601399 0.83 MEN1 (0.39) PDE4APDE4BPDE4CPDE4DSLC22A12
SCHEMBL8601274 0.83 PDE4A (0.46) PDE4APDE4BPDE4CPDE4DSLC22A12
SCHEMBL8601071 0.82 PDE4A (0.45) PDE4APDE4BPDE4CPDE4DPDE1A
SCHEMBL8600463 0.81 PDE4A (0.47) PDE4APDE4BPDE4CPDE4DSLC22A12
SCHEMBL8604472 0.81 PDE4A (0.47) PDE4APDE4BPDE4CPDE4DSLC22A12
SCHEMBL8601171 0.77 NR1D1 (0.40) PDE4APDE4BPDE4CPDE4DGAA
SCHEMBL8604717 0.76 PDE4A (0.46) PDE4APDE4BPDE4CPDE4DSLC22A12
SCHEMBL8603224 0.75 PDE4A (0.46) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL8600001 0.75 CNR1 (0.40) PDE4APDE4BPDE4CPDE4DTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998005327-A1 SUBSTITUTED AROMATIC COMPOUNDS RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1998-02-12 WO disclosed