SCHEMBL8601274

SCHEMBL8601274

Cc1cn(Cc2ccc3ccccc3c2)c2cc(C3CCNC3=O)ccc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 3/20 0.46
PDE4B Q07343 3/20 0.46
PDE4C Q08493 3/20 0.46
PDE4D Q08499 3/20 0.46
ICMT O60725 3/20 0.39
SLC5A1 P13866 1/20 0.37
SLC5A2 P31639 1/20 0.37
ACHE P22303 1/20 0.37
SLC22A12 Q96S37 3/20 0.36
BRD4 O60885 1/20 0.36
SLC6A2 P23975 2/20 0.36
SLC6A4 P31645 2/20 0.36
SLC6A3 Q01959 2/20 0.36
POLH Q9Y253 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
HDAC9 Q9UKV0 1/20 0.35
KCNH2 Q12809 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8599642 0.86 PDE4A (0.44) PDE4APDE4BPDE4CPDE4DSLC22A12
SCHEMBL8601071 0.85 PDE4A (0.45) PDE4APDE4BPDE4CPDE4DHDAC1
SCHEMBL8601399 0.85 MEN1 (0.39) PDE4APDE4BPDE4CPDE4DSLC22A12
SCHEMBL8601267 0.83 PDE4A (0.49) PDE4APDE4BPDE4CPDE4DSLC22A12
SCHEMBL8600463 0.82 PDE4A (0.47) PDE4APDE4BPDE4CPDE4DSLC22A12
SCHEMBL8604472 0.82 PDE4A (0.47) PDE4APDE4BPDE4CPDE4DICMT
SCHEMBL8601171 0.78 NR1D1 (0.40) PDE4APDE4BPDE4CPDE4DICMT
SCHEMBL8603224 0.76 PDE4A (0.46) PDE4APDE4BPDE4CPDE4D
SCHEMBL8649978 0.76 PDE4A (0.45) PDE4APDE4BPDE4CPDE4DICMT
SCHEMBL8601087 0.76 PDE4A (0.47) PDE4APDE4BPDE4CPDE4DBRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998005327-A1 SUBSTITUTED AROMATIC COMPOUNDS RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1998-02-12 WO disclosed