SCHEMBL8599642

SCHEMBL8599642

Cc1cn(Cc2ccc(Cl)cc2)c2cc(C3CCNC3=O)ccc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 6/20 0.44
PDE4B Q07343 6/20 0.44
PDE4C Q08493 6/20 0.44
PDE4D Q08499 6/20 0.44
SLC22A12 Q96S37 8/20 0.39
BRD4 O60885 2/20 0.36
KLK7 P49862 1/20 0.36
MAOA P21397 1/20 0.36
MAOB P27338 1/20 0.36
CACNB4 O00305 1/20 0.35
CACNA1A O00555 1/20 0.35
CACNA1G O43497 1/20 0.35
CACNG3 O60359 1/20 0.35
CACNA1F O60840 1/20 0.35
CACNA1H O95180 1/20 0.35
CACNB3 P54284 1/20 0.35
CACNA2D1 P54289 1/20 0.35
CACNG7 P62955 1/20 0.35
CACNA1B Q00975 1/20 0.35
CACNA1D Q01668 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8601399 0.91 MEN1 (0.39) PDE4APDE4BPDE4CPDE4DSLC22A12
SCHEMBL8604472 0.88 PDE4A (0.47) PDE4APDE4BPDE4CPDE4DSLC22A12
SCHEMBL8600463 0.88 PDE4A (0.47) PDE4APDE4BPDE4CPDE4DSLC22A12
SCHEMBL8601274 0.86 PDE4A (0.46) PDE4APDE4BPDE4CPDE4DSLC22A12
SCHEMBL8601267 0.84 PDE4A (0.49) PDE4APDE4BPDE4CPDE4DSLC22A12
SCHEMBL8601171 0.81 NR1D1 (0.40) PDE4APDE4BPDE4CPDE4D
SCHEMBL8603224 0.80 PDE4A (0.46) PDE4APDE4BPDE4CPDE4D
SCHEMBL8601087 0.79 PDE4A (0.47) PDE4APDE4BPDE4CPDE4DBRD4
SCHEMBL8600001 0.77 CNR1 (0.40) PDE4APDE4BPDE4CPDE4DBRD4
SCHEMBL8602159 0.76 BRD4 (0.41) PDE4APDE4BPDE4CPDE4DBRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998005327-A1 SUBSTITUTED AROMATIC COMPOUNDS RHONE-POULENC RORER PHARMACEUTICALS INC. (US) 1998-02-12 WO disclosed