SCHEMBL8604153

SCHEMBL8604153

CCCCOc1c(NC(C)C(C)C)c(=O)c1=O

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.39
ADAMTS5 Q9UNA0 2/20 0.37
CNR2 P34972 2/20 0.37
GAA P10253 2/20 0.33
PPARG P37231 2/20 0.32
PPARA Q07869 1/20 0.32
THRA P10827 1/20 0.32
THRB P10828 1/20 0.32
PLK1 P53350 1/20 0.32
MAPT P10636 2/20 0.31
MEN1 O00255 1/20 0.31
NPC1 O15118 1/20 0.31
ALDH1A1 P00352 1/20 0.31
RAB9A P51151 1/20 0.31
KMT2A Q03164 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7597268 0.84 PLK1 (0.43) POLBADAMTS5PLK1
SCHEMBL3717367 0.83 POLB (0.50) POLBGAAPLK1MAPTMEN1
SCHEMBL7604367 0.82 ADAMTS5 (0.38) POLBADAMTS5CNR2GAATHRA
SCHEMBL8598123 0.76 HDAC1 (0.36) POLBADAMTS5CNR2GAAMAPT
Squaric Acid Dibutyl Ester SCHEMBL56180 0.74 CYP3A4 (0.44) THRATHRBMAPTALDH1A1
SCHEMBL7597357 0.73 ADAMTS5 (0.38) POLBADAMTS5CNR2GAATHRA
SCHEMBL7602487 0.71 ADAMTS5 (0.37) POLBADAMTS5GAATHRATHRB
Squaric Acid Dibutyl Ester SCHEMBL2304620 0.70 THRA (0.36) POLBTHRATHRBMAPTALDH1A1
SCHEMBL9749015 0.70 CCNE2 (0.42) ADAMTS5GAAMAPTMEN1ALDH1A1
SCHEMBL9749261 0.70 ADAMTS5 (0.36) POLBADAMTS5GAATHRATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5763474-A SMOOTH MUSCLE RELAXANTS AMERICAN HOME PRODUCTS CORPORATION (US) 1998-06-09 US disclosed