SCHEMBL8604667

SCHEMBL8604667

CN1C(=O)CC(O)[C@@]2(C)C1CC[C@@H]1[C@H]2CC[C@]2(C)CCC[C@@H]12

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MBOAT4 Q96T53 3/20 0.42
NR1I3 Q14994 1/20 0.41
CDK5 Q00535 1/20 0.39
CDK5R1 Q15078 1/20 0.39
CYP19A1 P11511 3/20 0.39
AR P10275 1/20 0.38
GRIN1 Q05586 1/20 0.38
GRIN2B Q13224 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7741691 0.83 SRD5A2 (0.41) MBOAT4GRIN1GRIN2B
SCHEMBL8523823 0.82 AR (0.38) AR
SCHEMBL8523105 0.80 SHBG (0.36) MBOAT4NR1I3ARGRIN1GRIN2B
SCHEMBL7711769 0.80 MBOAT4 (0.38) MBOAT4CDK5CDK5R1CYP19A1GRIN1
SCHEMBL27369735 0.80 MBOAT4 (0.39) MBOAT4CDK5CDK5R1CYP19A1GRIN1
SCHEMBL5596628 0.80 SRD5A1 (0.54)
SCHEMBL4729968 0.80 SRD5A1 (0.54)
SCHEMBL8713486 0.79 SRD5A1 (0.41) MBOAT4GRIN1GRIN2B
SCHEMBL8528297 0.78 HSD17B7 (0.42) MBOAT4
SCHEMBL8823339 0.78 MBOAT4 (0.38) MBOAT4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786999-A4 COMBINATION METHOD FOR ACNE TREATMENT MERCK & CO INC (US) 1999-01-20 EP disclosed
EP-0792371-A4 COMBINATION METHOD FOR ACNE TREATMENT MERCK & CO INC (US) 1998-12-30 EP disclosed
EP-0792371-A1 COMBINATION METHOD FOR ACNE TREATMENT Merck & Co., Inc. (US) 1997-09-03 EP disclosed
EP-0786999-A1 COMBINATION METHOD FOR ACNE TREATMENT Merck & Co., Inc. (US) 1997-08-06 EP disclosed
WO-1996012487-A1 COMBINATION METHOD FOR ACNE TREATMENT MERCK & CO., INC. (US) 1996-05-02 WO disclosed
WO-1996012817-A1 COMBINATION METHOD FOR ACNE TREATMENT MERCK & CO., INC. (US) 1996-05-02 WO disclosed