SCHEMBL8606451

SCHEMBL8606451

CC(C)(Oc1ccc(Cl)cc1)c1ccn2ncnc2n1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 5/20 0.34
CYP3A4 P08684 4/20 0.34
KDM4E B2RXH2 3/20 0.34
CYP1A2 P05177 3/20 0.34
MEN1 O00255 2/20 0.34
MAPT P10636 2/20 0.34
CYP2C19 P33261 2/20 0.34
KMT2A Q03164 2/20 0.34
CYP2D6 P10635 1/20 0.34
ALDH1A1 P00352 3/20 0.34
TSHR P16473 3/20 0.34
PPARG P37231 2/20 0.33
FABP2 P12104 1/20 0.33
SLC22A12 Q96S37 1/20 0.33
POLB P06746 1/20 0.33
HSP90AA1 P07900 1/20 0.33
HPGD P15428 2/20 0.32
SCN5A Q14524 1/20 0.32
KIT P10721 3/20 0.31
PDE10A Q9Y233 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12603986 0.75 ALDH1A1 (0.42) KDM4EMEN1CYP2C19KMT2AALDH1A1
SCHEMBL8605894 0.71 L3MBTL1 (0.39) CYP3A4KDM4ECYP1A2MEN1CYP2C19
SCHEMBL7552061 0.69 ALDH1A1 (0.44) PPARACYP3A4KDM4ECYP1A2MEN1
SCHEMBL22109267 0.69 KDM4E (0.38) KDM4EALDH1A1PDE10AMAPK1
SCHEMBL8606554 0.68 KDM4E (0.32) CYP3A4KDM4EMAPTALDH1A1POLB
SCHEMBL8607084 0.63 SCN5A (0.42) KDM4EMAPTALDH1A1POLBSCN5A
SCHEMBL2492473 0.63 ALDH1A1 (0.46) KDM4ECYP1A2MEN1MAPTKMT2A
SCHEMBL4820655 0.62 PPARA (0.55) PPARACYP3A4CYP1A2MEN1MAPT
SCHEMBL18676744 0.60 MAOA (0.42) PPARACYP3A4KDM4ECYP1A2MEN1
SCHEMBL9933093 0.60 PDE10A (0.45) KDM4ECYP2C19ALDH1A1PDE10AMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753665-A TRIAZOLOPYRIMIDINES, NERVOUS SYSTEM DISORDERS KNOLL AKTIENGESELLSCHAFT (DE) 1998-05-19 US claimed
US-5753665-A TRIAZOLOPYRIMIDINES, NERVOUS SYSTEM DISORDERS KNOLL AKTIENGESELLSCHAFT (DE) 1998-05-19 US disclosed