SCHEMBL860866

SCHEMBL860866

Clc1cccc2c1=C1CN(Cc3ccccc3)CC1CNC=2

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 6/20 0.37
DRD2 P14416 1/20 0.36
DRD4 P21917 1/20 0.36
DRD3 P35462 1/20 0.36
ESR1 P03372 1/20 0.36
ESR2 Q92731 1/20 0.36
FUCA1 P04066 2/20 0.35
DPP4 P27487 1/20 0.34
S1PR1 P21453 1/20 0.34
S1PR5 Q9H228 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL861661 0.81 SIGMAR1 (0.42) SIGMAR1DRD2DRD4DRD3ESR1
SCHEMBL2598136 0.74 BRD4 (0.41) SIGMAR1DRD2DRD4DRD3MEN1
SCHEMBL861689 0.74 DRD2 (0.38) SIGMAR1DRD2DRD4DRD3FUCA1
Hydrochloric Acid SCHEMBL2268301 0.72 SIGMAR1 (0.43) SIGMAR1DRD4FUCA1MEN1KMT2A
SCHEMBL24326131 0.59 ALDH1A1 (0.50) SIGMAR1ESR1ESR2FUCA1S1PR1
SCHEMBL477142 0.58 FUCA1 (0.55) SIGMAR1DRD2DRD3FUCA1S1PR1
SCHEMBL4279682 0.58 FUCA1 (0.55) SIGMAR1FUCA1S1PR1S1PR5MEN1
SCHEMBL3522693 0.58 FUCA1 (0.55) SIGMAR1FUCA1S1PR1S1PR5MEN1
SCHEMBL3522692 0.58 FUCA1 (0.55) SIGMAR1FUCA1S1PR1S1PR5MEN1
SCHEMBL3324661 0.58 FUCA1 (0.55) SIGMAR1FUCA1S1PR1S1PR5MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2432783-A1 MODULATORS OF 5-HT RECEPTORS AND METHODS OF USE THEREOF Abbott Laboratories (US) 2012-03-28 EP disclosed
WO-2010135560-A1 MODULATORS OF 5-HT RECEPTORS AND METHODS OF USE THEREOF ABBOTT LABORATORIES (US) 2010-11-25 WO disclosed