SCHEMBL861689

SCHEMBL861689

Fc1ccc2c(c1)=C1CN(Cc3ccccc3)CC1CNC=2

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.38
DRD3 P35462 1/20 0.38
ACHE P22303 8/20 0.38
BACE1 P56817 7/20 0.37
BCHE P06276 5/20 0.37
TACR1 P25103 2/20 0.37
DRD4 P21917 1/20 0.37
FUCA1 P04066 2/20 0.36
SIGMAR1 Q99720 1/20 0.36
CCR5 P51681 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL861661 0.83 SIGMAR1 (0.42) DRD2DRD3DRD4FUCA1SIGMAR1
SCHEMBL860866 0.74 SIGMAR1 (0.37) DRD2DRD3DRD4FUCA1SIGMAR1
SCHEMBL2598136 0.70 BRD4 (0.41) DRD2DRD3BCHEDRD4SIGMAR1
Hydrochloric Acid SCHEMBL2268301 0.70 SIGMAR1 (0.43) ACHEDRD4FUCA1SIGMAR1
SCHEMBL4404973 0.64 DRD2 (0.55) DRD2DRD3ACHEBACE1BCHE
SCHEMBL4224135 0.62 SIGMAR1 (0.55) DRD2DRD3ACHEBACE1BCHE
SCHEMBL8725812 0.62 SIGMAR1 (0.75) ACHEBACE1BCHESIGMAR1
SCHEMBL16225922 0.62 ALDH1A1 (0.74) SIGMAR1
SCHEMBL16226988 0.60 ACHE (0.69) ACHEBACE1BCHESIGMAR1
SCHEMBL16227202 0.60 SIGMAR1 (0.60) ACHEBACE1BCHESIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2432783-A1 MODULATORS OF 5-HT RECEPTORS AND METHODS OF USE THEREOF Abbott Laboratories (US) 2012-03-28 EP disclosed
WO-2010135560-A1 MODULATORS OF 5-HT RECEPTORS AND METHODS OF USE THEREOF ABBOTT LABORATORIES (US) 2010-11-25 WO disclosed