SCHEMBL860949

SCHEMBL860949

O=C(OCc1ccccc1)[C@H](CC1CCC1)N(Cc1ccccc1)Cc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
ATM Q13315 1/20 0.44
CTSL P07711 1/20 0.43
CTSB P07858 1/20 0.43
CTSS P25774 1/20 0.43
CTSK P43235 1/20 0.43
EPOR P19235 2/20 0.42
TSHR P16473 1/20 0.41
ALDH1A1 P00352 3/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ENPP2 Q13822 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
MAPK1 P28482 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A3 Q01959 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL840766 0.85 ATM (0.48) ATMALDH1A1NPC1RAB9AMAPK1
SCHEMBL841071 0.85 ATM (0.48) ATMALDH1A1NPC1RAB9AMAPK1
SCHEMBL878904 0.84 ATM (0.45) CYP3A4ATMCTSKEPORTSHR
SCHEMBL9076431 0.83 ATM (0.51) ATMCTSLCTSBCTSSCTSK
SCHEMBL9076426 0.83 ATM (0.51) ATMCTSLCTSBCTSSCTSK
SCHEMBL9076021 0.81 ATM (0.53) ATMALDH1A1NPC1RAB9ASMN1; SMN2
SCHEMBL9076016 0.81 ATM (0.53) ATMALDH1A1NPC1RAB9ASMN1; SMN2
SCHEMBL8059476 0.80 CYP2C19 (0.50) CYP3A4CYP2C9CYP2C19CTSLCTSB
SCHEMBL20858214 0.79 EPOR (0.49) CYP3A4CYP2C9CYP2C19EPORALDH1A1
SCHEMBL7438541 0.79 CTRB1 (0.49) CTSBEPORALDH1A1L3MBTL1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143448-B2 Process for the preparation of (3S)-3-amino-N-cyclopropyl-2-hydroxyalkanamide derivatives VIROBAY, INC. (US) 2012-03-27 US disclosed
US-20090312571-A1 PROCESS FOR THE PREPARATION OF (3S)-3-AMINO-N-CYCLOPROPYL-2-HYDROXYALKANAMIDE DERIVATIVES VIROBAY, INC. (US) 2009-12-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090312571-A1 PROCESS FOR THE PREPARATION OF (3S)-3-AMINO-N-CYCLOPROPYL-2-HYDROXYALKANAMIDE DERIVATIVES HCN3, NPEPPS, HACL2 CYP3A4 432/4885CYP2C9 811/4885CYP2C19 1327/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.