SCHEMBL8610348

SCHEMBL8610348

CC1(c2c[nH]cn2)Cc2ccc(F)cc2C1=O

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 5/20 0.36
ACHE P22303 1/20 0.35
PARP1 P09874 1/20 0.35
PARP10 Q53GL7 1/20 0.35
SRD5A1 P18405 2/20 0.35
TYMS P04818 1/20 0.34
CHRM1 P11229 1/20 0.33
HRH1 P35367 1/20 0.33
PAK1 Q13153 1/20 0.33
CYP1A2 P05177 1/20 0.33
MAPT P10636 1/20 0.33
CYP2C19 P33261 1/20 0.33
KMT2A Q03164 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA7 P43166 1/20 0.33
CA9 Q16790 1/20 0.33
ALPL P05186 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8614404 0.84 CYP19A1 (0.35) PARP1TYMSKMT2ACA9
SCHEMBL7639950 0.81 ADRA2A (0.37) AKR1B1ACHEPARP1PARP10SRD5A1
SCHEMBL8616201 0.81 KDM4E (0.39) MAPT
SCHEMBL7645070 0.75 ADRA2A (0.42) AKR1B1SRD5A1
SCHEMBL2390689 0.75 ACHE (0.46) AKR1B1ACHEPARP1PARP10SRD5A1
Fipamezole SCHEMBL935549 0.69 ADRA2A (0.57)
Fipamezole SCHEMBL1271449 0.69 ADRA2A (0.57)
Fipamezole SCHEMBL3901401 0.68 ADRA2A (0.56)
SCHEMBL24376604 0.67 CA1 (0.44) AKR1B1ACHEPARP1PARP10SRD5A1
SCHEMBL8611882 0.66 ALDH1A1 (0.39) AKR1B1ACHEMAPTCYP2C19KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0618906-B1 SUBSTITUTED IMIDAZOLE DERIVATIVES AND THEIR PREPARATION AND USE JUVANTIA PHARMA LTD OY (FI) 1998-04-22 EP disclosed
US-5498623-A MULTISTAGE REACTION FOR HALOGENATION OF COMPOUNDS, NITRATION, REDUCTION AND CONVERSION TO DIAZONIUM SALT THEN HALOGENATION FOR COGNITIVE DISORDERS ORION-YHTYMA OY (FI) 1996-03-12 US disclosed
EP-0618906-A1 SUBSTITUTED IMIDAZOLE DERIVATIVES AND THEIR PREPARATION AND USE ANTII SAKARI HAAPALINNA (FI) 1994-10-12 EP disclosed
WO-1993013074-A1 SUBSTITUTED IMIDAZOLE DERIVATIVES AND THEIR PREPARATION AND USE Orion-Yhtymä Oy (FI) 1993-07-08 WO disclosed