SCHEMBL8611882

SCHEMBL8611882

CCC1(c2c[nH]cn2)Cc2ccc([N+](=O)[O-])cc2C1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.39
TDP2 O95551 1/20 0.39
CAPN9 O14815 1/20 0.39
CASP3 P42574 1/20 0.39
CYP3A4 P08684 2/20 0.38
TDP1 Q9NUW8 1/20 0.38
ADRA2A P08913 1/20 0.37
PNMT P11086 1/20 0.37
ADRA2B P18089 1/20 0.37
ADRA2C P18825 1/20 0.37
AKR1B1 P15121 1/20 0.37
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
ACHE P22303 4/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8611842 0.83 ALDH1A1 (0.42) ALDH1A1TDP2CAPN9CASP3CYP3A4
SCHEMBL8611233 0.82 CYP19A1 (0.39) CYP3A4CA9PDE4D
SCHEMBL8614549 0.82 AKR1B1 (0.34) AKR1B1ACHEMAPT
SCHEMBL8610413 0.79 NPSR1 (0.43) ALDH1A1TDP2MEN1KMT2AMAPT
SCHEMBL8613817 0.79 PNMT (0.41) TDP2CYP3A4ADRA2APNMTADRA2B
SCHEMBL8610780 0.76 PNMT (0.43) TDP2CYP3A4ADRA2APNMTADRA2B
SCHEMBL9139518 0.72 CA1 (0.50) ALDH1A1TDP2CAPN9CASP3CYP3A4
SCHEMBL9431991 0.70 NPSR1 (0.40) ALDH1A1TDP2MEN1KMT2AMAPT
SCHEMBL8614404 0.66 CYP19A1 (0.35) TDP2TDP1CA9KMT2A
SCHEMBL23674967 0.65 SIRT2 (0.44) ALDH1A1TDP2CAPN9CASP3CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0618906-B1 SUBSTITUTED IMIDAZOLE DERIVATIVES AND THEIR PREPARATION AND USE JUVANTIA PHARMA LTD OY (FI) 1998-04-22 EP disclosed
US-5498623-A MULTISTAGE REACTION FOR HALOGENATION OF COMPOUNDS, NITRATION, REDUCTION AND CONVERSION TO DIAZONIUM SALT THEN HALOGENATION FOR COGNITIVE DISORDERS ORION-YHTYMA OY (FI) 1996-03-12 US disclosed
EP-0618906-A1 SUBSTITUTED IMIDAZOLE DERIVATIVES AND THEIR PREPARATION AND USE ANTII SAKARI HAAPALINNA (FI) 1994-10-12 EP disclosed
WO-1993013074-A1 SUBSTITUTED IMIDAZOLE DERIVATIVES AND THEIR PREPARATION AND USE Orion-Yhtymä Oy (FI) 1993-07-08 WO disclosed