SCHEMBL8614404

SCHEMBL8614404

CC1(c2c[nH]cn2)Cc2ccc(N)cc2C1=O

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.35
CA9 Q16790 1/20 0.33
TYMS P04818 1/20 0.33
PARP1 P09874 2/20 0.31
TDP2 O95551 1/20 0.31
CRBN Q96SW2 2/20 0.30
DDB1 Q16531 1/20 0.30
KDM4E B2RXH2 1/20 0.30
GAA P10253 1/20 0.30
APEX1 P27695 1/20 0.30
KMT2A Q03164 1/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8610348 0.84 AKR1B1 (0.36) CA9TYMSPARP1KMT2A
SCHEMBL8611233 0.81 CYP19A1 (0.39) CYP19A1CA9TYMS
SCHEMBL8616201 0.81 KDM4E (0.39) TDP2KDM4EGAA
SCHEMBL8613975 0.75 KDM4E (0.30) CA9KDM4EGAAAPEX1KMT2A
SCHEMBL9140465 0.75 CA9 (0.40) CYP19A1CA9TYMSPARP1TDP2
SCHEMBL8610304 0.69 ADRA2A (0.40) CYP19A1
SCHEMBL27463810 0.66 CA9 (0.41) CA9TYMSPARP1TDP2CRBN
SCHEMBL8611882 0.66 ALDH1A1 (0.39) CA9TDP2KMT2ATDP1
SCHEMBL8614549 0.66 AKR1B1 (0.34) TYMSPARP1
SCHEMBL1709821 0.63 CA9 (0.53) CYP19A1CA9TDP2KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0618906-B1 SUBSTITUTED IMIDAZOLE DERIVATIVES AND THEIR PREPARATION AND USE JUVANTIA PHARMA LTD OY (FI) 1998-04-22 EP disclosed
US-5498623-A MULTISTAGE REACTION FOR HALOGENATION OF COMPOUNDS, NITRATION, REDUCTION AND CONVERSION TO DIAZONIUM SALT THEN HALOGENATION FOR COGNITIVE DISORDERS ORION-YHTYMA OY (FI) 1996-03-12 US disclosed