SCHEMBL8611233

SCHEMBL8611233

CCC1(c2c[nH]cn2)Cc2ccc(N)cc2C1=O

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 7/20 0.39
CYP3A4 P08684 2/20 0.35
CYP17A1 P05093 1/20 0.35
CYP11A1 P05108 1/20 0.35
TBXAS1 P24557 1/20 0.35
PMP22 Q01453 1/20 0.35
PDE4D Q08499 1/20 0.35
PDE3A Q14432 1/20 0.35
NFKB1 P19838 1/20 0.35
NPSR1 Q6W5P4 1/20 0.32
CA9 Q16790 1/20 0.31
TYMS P04818 1/20 0.31
RET P07949 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8614549 0.85 AKR1B1 (0.34) TYMS
SCHEMBL7639950 0.85 ADRA2A (0.37) CA9TYMS
SCHEMBL8611882 0.82 ALDH1A1 (0.39) CYP3A4PDE4DCA9
SCHEMBL8610413 0.82 NPSR1 (0.43) NPSR1
SCHEMBL8614404 0.81 CYP19A1 (0.35) CYP19A1CA9TYMS
SCHEMBL8610304 0.74 ADRA2A (0.40) CYP19A1
SCHEMBL9431991 0.72 NPSR1 (0.40) CYP19A1NPSR1
SCHEMBL8613975 0.70 KDM4E (0.30) CA9
SCHEMBL9140465 0.66 CA9 (0.40) CYP19A1CYP3A4NPSR1CA9TYMS
SCHEMBL8610348 0.66 AKR1B1 (0.36) CA9TYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0618906-B1 SUBSTITUTED IMIDAZOLE DERIVATIVES AND THEIR PREPARATION AND USE JUVANTIA PHARMA LTD OY (FI) 1998-04-22 EP disclosed
US-5498623-A MULTISTAGE REACTION FOR HALOGENATION OF COMPOUNDS, NITRATION, REDUCTION AND CONVERSION TO DIAZONIUM SALT THEN HALOGENATION FOR COGNITIVE DISORDERS ORION-YHTYMA OY (FI) 1996-03-12 US disclosed
EP-0618906-A1 SUBSTITUTED IMIDAZOLE DERIVATIVES AND THEIR PREPARATION AND USE ANTII SAKARI HAAPALINNA (FI) 1994-10-12 EP disclosed
WO-1993013074-A1 SUBSTITUTED IMIDAZOLE DERIVATIVES AND THEIR PREPARATION AND USE Orion-Yhtymä Oy (FI) 1993-07-08 WO disclosed